SCHEMBL361027

SCHEMBL361027

CON(C)C(=O)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.53
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
AKR1B1 P15121 1/20 0.48
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
HDAC4 P56524 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
LTB4R Q15722 3/20 0.47
LTB4R2 Q9NPC1 3/20 0.47
TRPM8 Q7Z2W7 1/20 0.46
TSHR P16473 1/20 0.46
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 1/20 0.44
LMNA P02545 1/20 0.44
REN P00797 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1515926 0.90 LMNA (0.55) ALOX5HDAC4HDAC6TSHRALDH1A1
SCHEMBL2353230 0.86 ALOX5 (0.76) ALOX5NPC1RAB9ALTB4RLTB4R2
SCHEMBL1515761 0.85 AOC3 (0.54) LTB4RLTB4R2
SCHEMBL4952728 0.85 FFAR1 (0.58) ALOX5HDAC4HDAC6LTB4RLTB4R2
SCHEMBL9903521 0.84 RAB9A (0.45) ALOX5CES2CES1AKR1B1NPC1
SCHEMBL8064820 0.83 HDAC4 (0.49) ALOX5NPC1RAB9AHDAC4HDAC6
SCHEMBL13226836 0.83 HDAC4 (0.49) ALOX5HDAC4HDAC6ALDH1A1SMN1; SMN2
SCHEMBL8371453 0.83 HDAC4 (0.49) ALOX5HDAC4HDAC6LTB4RLTB4R2
SCHEMBL1058423 0.82 CTBP2 (0.50) NPC1RAB9ALTB4RLTB4R2ALDH1A1
SCHEMBL12570225 0.82 NPC1 (0.51) NPC1RAB9AHDAC6ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 212 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026101698-A1 HEPCIDIN MIMETIC COMPOUNDS AND USES THEREOF PROTAGONIST THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
WO-2025262192-A1 QUINAZOLINE DERIVATIVES SUITABLE FOR USE AS WERNER SYNDROME HELICASE PROTEIN INHIBITORS BREAKPOINT THERAPEUTICS GMBH (DE) 2025-12-26 WO disclosed
CN-114269720-B Acetyl-coa synthetase short chain2(ACSS2) Small molecule inhibitors of (a) 库拉德夫制药私人有限公司 2025-03-28 CN disclosed
CN-113801163-B Organic arsenic-based II-type pyruvate kinase inhibitor and preparation method and application thereof 中国科学院上海有机化学研究所 2025-03-04 CN disclosed
US-11918656-B2 Antibody-drug-conjugate and its use for the treatment of cancer PIERRE FABRE MEDICAMENT (FR) 2024-03-05 US disclosed
US-20230331707-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2023-10-19 US disclosed
US-20230331707-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2023-10-19 US disclosed
US-20230331707-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF SHANGHAI INSTITUTE OF ORGANIC CHEMISTRY, CHINESE ACADEMY OF SCIENCES (CN) 2023-10-19 US disclosed
CN-116514679-A Palladium-catalyzed sp with low-cost and high-efficiency quaternary ammonium nitrate as oxidant 2 And sp (sp) 3 Carbon hydrogen bond alkenylation method 南京工业大学 2023-08-01 CN disclosed
US-20230234917-A1 ASPARAGINE DERIVATIVES AND METHODS OF USING SAME SENDA BIOSCIENCES INC (US) 2023-07-27 US disclosed
WO-2001055096-A1 METHOD FOR PRODUCING N-ALKOXY-N-ALKYLAMIDES LONZA AG (CH) 2001-08-02 WO disclosed
EP-1091938-A2 ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF Aventis Pharmaceuticals Inc. (US) 2001-04-18 EP disclosed
EP-0971894-A1 NICOTINAMIDE DERIVATIVES Pfizer Products Inc. (US) 2000-01-19 EP disclosed
WO-2000001671-A2 ANTIHISTAMINIC PIPERIDINE DERIVATIVES AND INTERMEDIATES FOR THE PREPARATION THEREOF AVENTIS PHARMACEUTICALS INC. (US) 2000-01-13 WO disclosed
WO-1998045268-A1 NICOTINAMIDE DERIVATIVES PFIZER PRODUCTS INC. (US) 1998-10-15 WO disclosed
US-5691356-A ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 1997-11-25 US disclosed
EP-0772601-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1997-05-14 EP disclosed
WO-1996003387-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed
EP-0388691-A1 Azole-1-alkanamides as antiarrhytmic agents and preparation thereof STERLING DRUG INC. (US) 1990-09-26 EP disclosed
US-4925857-A Pyridinyl-1H-pyrazole-1-alkanamides as antiarrhythmic agents STERLING DRUG INC. (US) 1990-05-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230331707-A1 PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF RIPK1, RIPK4, RIPK3 ALOX5 2183/4885CES2 4869/4885CES1 2783/4885
US-11918656-B2 Antibody-drug-conjugate and its use for the treatment of cancer DDOST, DAD1, KRTCAP2 ALOX5 1177/4885CES2 2739/4885CES1 820/4885
US-20230234917-A1 ASPARAGINE DERIVATIVES AND METHODS OF USING SAME ASNS, SI, NARS1 ALOX5 1486/4885CES2 2523/4885CES1 954/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.