SCHEMBL363071

SCHEMBL363071

Cc1cc(/C(CC(c2ccc(C(=O)NCC(F)(F)F)c(F)c2)c2ccccc2Cl)=N/O)c[nH]c1=O

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.37
OPRD1 P41143 1/20 0.36
HSD17B2 P37059 2/20 0.34
GPBAR1 Q8TDU6 3/20 0.33
F9 P00740 4/20 0.33
P2RX7 Q99572 1/20 0.33
S1PR1 P21453 1/20 0.32
S1PR3 Q99500 1/20 0.32
MCL1 Q07820 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
PPARG P37231 1/20 0.31
HTRA1 Q92743 1/20 0.30
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364487 0.92 BRD4 (0.42) BRD4HSD17B2GPBAR1F9S1PR1
SCHEMBL364524 0.89 PTGS2 (0.36) BRD4GPBAR1F9CTSA
SCHEMBL361665 0.86 HPGD (0.37) BRD4GPBAR1
SCHEMBL362599 0.84 BRD4 (0.40) BRD4GPBAR1
SCHEMBL362147 0.84 MET (0.34) BRD4GPBAR1F9
SCHEMBL363606 0.84 GPBAR1 (0.35) BRD4GPBAR1
SCHEMBL364618 0.83 MET (0.42) BRD4GPBAR1P2RX7
SCHEMBL1389788 0.82 OPRD1 (0.37) BRD4OPRD1HSD17B2GPBAR1F9
SCHEMBL1389780 0.82 OPRD1 (0.37) BRD4OPRD1HSD17B2GPBAR1F9
SCHEMBL1389785 0.82 OPRD1 (0.37) BRD4OPRD1HSD17B2GPBAR1F9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP claimed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO claimed
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed