SCHEMBL366133

SCHEMBL366133

CN(C)CCS(=O)(=O)c1ccc2c(C(=O)O)c3ccccc3n2c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.41
HTR6 P50406 13/20 0.40
HTR1A P08908 1/20 0.40
DRD2 P14416 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR1F P30939 1/20 0.40
HTR7 P34969 1/20 0.40
DRD3 P35462 1/20 0.40
TNF P01375 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL364606 0.90 HTR6 (0.38) AGTR1HTR6HTR1ADRD2HTR1D
SCHEMBL365522 0.88 MEN1 (0.41) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL366693 0.86 ALDH1A1 (0.47) HTR6HTR1ADRD2HTR1DHTR1B
SCHEMBL366132 0.82 ALDH1A1 (0.38) AGTR1HTR6HTR1ADRD2HTR1D
SCHEMBL366462 0.82 LMNA (0.46) AGTR1
SCHEMBL367747 0.80 AGTR1 (0.48) AGTR1
SCHEMBL365648 0.77 CA9 (0.45) AGTR1
SCHEMBL366536 0.74 EGFR (0.53)
SCHEMBL366858 0.74 KMT2A (0.43)
SCHEMBL365147 0.73 AGTR1 (0.39) AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed