SCHEMBL367389

SCHEMBL367389

O=C(O)c1c2c(O)cc(OS(=O)(=O)C3CC3)cc2n2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.36
PTGS2 P35354 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
APAF1 O14727 1/20 0.32
MAPT P10636 1/20 0.32
G6PD P11413 1/20 0.32
PABPC1 P11940 1/20 0.32
CACNA1B Q00975 1/20 0.32
APBA1 Q02410 1/20 0.32
KMT2A Q03164 1/20 0.32
SAE1 Q9UBE0 1/20 0.32
UBA2 Q9UBT2 1/20 0.32
RORC P51449 1/20 0.31
BAZ2B Q9UIF8 1/20 0.30
BAZ2A Q9UIF9 1/20 0.30
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL367244 0.90 KDM4E (0.33) IDO1ALDH1A1KDM4EMEN1APAF1
SCHEMBL365225 0.86 CA12 (0.35) IDO1PTGS2ALDH1A1KDM4EMEN1
SCHEMBL366115 0.86 CA1 (0.41) IDO1PTGS2ALDH1A1KDM4EMEN1
SCHEMBL366074 0.77 POLB (0.33) IDO1ALDH1A1KDM4EMEN1APAF1
SCHEMBL365406 0.77 STS (0.39) ALDH1A1KDM4EMEN1APAF1MAPT
SCHEMBL367408 0.74 EPHX1 (0.51) KDM4EMEN1KMT2ACYP1A2
SCHEMBL365212 0.74 KMT2A (0.39) IDO1PTGS2ALDH1A1KDM4EMEN1
SCHEMBL367390 0.74 AGTR1 (0.34) ALDH1A1KDM4EMEN1MAPTKMT2A
SCHEMBL367670 0.73 ALDH1A1 (0.40) IDO1PTGS2ALDH1A1KDM4EMEN1
SCHEMBL366019 0.73 STS (0.41) IDO1PTGS2ALDH1A1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed