SCHEMBL3639293

SCHEMBL3639293

CCOC(=O)n1c(C(=O)O)cc2cc(NC(C)=O)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.47
KMT2A Q03164 3/20 0.45
MEN1 O00255 2/20 0.45
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.43
MAPT P10636 2/20 0.42
NPC1 O15118 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
RORC P51449 1/20 0.41
TP53 P04637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LMNA P02545 3/20 0.41
ADORA3 P0DMS8 1/20 0.41
F2 P00734 1/20 0.41
PLAU P00749 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13560521 0.86 ECE1 (0.39) MMP13KMT2AMEN1SMN1; SMN2KDM4E
SCHEMBL3639291 0.84 MMP13 (0.52) MMP13KMT2AMEN1CYP2C19SMN1; SMN2
SCHEMBL3036607 0.82 MMP13 (0.47) MMP13KMT2AMEN1CYP2C19SMN1; SMN2
SCHEMBL3637426 0.80 ABCB11 (0.45) KMT2AMEN1SMN1; SMN2KDM4EALDH1A1
SCHEMBL13560519 0.77 TSPO (0.38) MMP13KMT2AMEN1SMN1; SMN2ALDH1A1
SCHEMBL3638010 0.75 CCR2 (0.50) KMT2AMEN1SMN1; SMN2ALDH1A1MAPT
SCHEMBL3675353 0.72 KDM4E (0.42) KMT2AMEN1SMN1; SMN2KDM4EALDH1A1
SCHEMBL3639124 0.72 SRD5A2 (0.69) KMT2AMEN1KDM4EALDH1A1NPC1
SCHEMBL3641237 0.72 ACSS2 (0.38) KMT2AMEN1SMN1; SMN2KDM4EALDH1A1
SCHEMBL3634758 0.71 SRD5A2 (0.44) KMT2AMEN1SMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2166856-A1 CHEMICAL COMPOUNDS GlaxoSmithKline LLC (US) 2010-03-31 EP disclosed
WO-2008154271-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2008-12-18 WO disclosed