SCHEMBL367705

SCHEMBL367705

CSc1ccc2c(C(N)=O)c3ccccc3n2c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.48
SRC P12931 5/20 0.48
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
BRCA1 P38398 1/20 0.35
NR4A2 P43354 1/20 0.33
AGTR1 P30556 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365779 0.87 EGFR (0.43) EGFRSRCALDH1A1POLBKDM4E
SCHEMBL365370 0.83 NPC1 (0.47) EGFRSRCALDH1A1KDM4EMEN1
SCHEMBL367201 0.79 EGFR (0.45) EGFRSRCHTR2AHTR2CALDH1A1
SCHEMBL367764 0.79 EGFR (0.45) EGFRSRCHTR2AHTR2CALDH1A1
SCHEMBL367704 0.79 EGFR (0.43) EGFRSRCALDH1A1POLBKDM4E
SCHEMBL367330 0.78 EGFR (0.46) EGFRSRCHTR2AHTR2CALDH1A1
SCHEMBL367707 0.77 EGFR (0.44) EGFRSRCHTR2AHTR2CMEN1
SCHEMBL364594 0.77 EGFR (0.44) EGFRSRCALDH1A1POLBKDM4E
SCHEMBL365259 0.77 KDM4E (0.44) EGFRSRCHTR2AHTR2CALDH1A1
SCHEMBL367114 0.76 ALDH1A1 (0.49) EGFRSRCALDH1A1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO claimed
WO-2012007008-A1 INHIBITORS OF HDME EPITHERAPEUTICS APS (DK) 2012-01-19 WO disclosed