SCHEMBL370096

SCHEMBL370096

CC(=O)Nc1cccc(C(CC(=NO)C2=CC=CN(C)C2)c2ccc(Cl)cc2F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.36
HPGD P15428 1/20 0.34
MCHR1 Q99705 2/20 0.34
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
CMA1 P23946 1/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
SLC6A3 Q01959 2/20 0.33
KCNH2 Q12809 2/20 0.33
POLB P06746 1/20 0.33
HDAC1 Q13547 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL368192 0.80 CREBBP (0.40) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL368191 0.80 CREBBP (0.40) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL368193 0.80 CREBBP (0.40) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL363191 0.76 ALDH1A1 (0.38) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL370503 0.73 GPBAR1 (0.46) MEN1KMT2A
SCHEMBL370370 0.72 FFAR1 (0.33)
SCHEMBL1390327 0.72 CREBBP (0.42) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2
SCHEMBL370694 0.71 GPBAR1 (0.37) ALDH1A1MEN1KMT2ASMN1; SMN2CYP2D6
SCHEMBL369976 0.70 GPBAR1 (0.35) ALDH1A1POLB
SCHEMBL364598 0.68 ALDH1A1 (0.38) ALDH1A1MAPTMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed