SCHEMBL3704897

SCHEMBL3704897

CCCNc1ccc(-c2ccccc2)c(C)c1C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
ALDH1A1 P00352 5/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
KDM4E B2RXH2 4/20 0.38
HPGD P15428 4/20 0.38
HSD17B10 Q99714 1/20 0.38
PLA2G1B P04054 1/20 0.37
BCAT2 O15382 1/20 0.37
HTT P42858 2/20 0.37
LMNA P02545 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.37
SOAT1 P35610 2/20 0.36
KDM6B O15054 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
HCAR3 P49019 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ABCB1 P08183 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3708760 0.92 KDM4E (0.47) ALDH1A1MEN1KMT2APOLBKDM4E
SCHEMBL3698514 0.89 FABP4 (0.40) IDO1ALDH1A1MEN1KMT2APOLB
SCHEMBL3714028 0.84 ALDH1A1 (0.46) IDO1ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL3135452 0.75 BCAT2 (0.47) ALDH1A1MEN1KMT2APOLBKDM4E
SCHEMBL3701694 0.73 BCAT2 (0.46) ALDH1A1MEN1KMT2APOLBHPGD
Hydrochloric Acid SCHEMBL29287793 0.73 CA1 (0.47) ALDH1A1MEN1KMT2APOLBKDM4E
Hydrochloric Acid SCHEMBL29287828 0.73 CA1 (0.47) ALDH1A1MEN1KMT2APOLBKDM4E
SCHEMBL28568958 0.72 HSP90AA1 (0.46) PDCD1CD274
SCHEMBL28568956 0.72 HSP90AA1 (0.46) PDCD1CD274
SCHEMBL3704899 0.71 PARP1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2197835-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS Prosidion Limited (GB) 2010-06-23 EP disclosed
WO-2009030962-A1 BICYCLIC ARYL AND HETEROARYL RECEPTOR MODULATORS PROSIDION LIMITED (GB) 2009-03-12 WO disclosed