SCHEMBL3708634

SCHEMBL3708634

CCOC(=O)N(c1ccccc1Cl)c1c(C)noc1-c1ccc(COc2ccc(CC(=O)OC)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
ALOX5 P09917 5/20 0.40
ALOX5AP P20292 3/20 0.40
PPARD Q03181 5/20 0.39
ESR1 P03372 2/20 0.39
THRA P10827 2/20 0.39
THRB P10828 2/20 0.39
VDR P11473 2/20 0.39
RXRA P19793 2/20 0.39
PPARG P37231 2/20 0.39
PPARA Q07869 2/20 0.39
ESR2 Q92731 2/20 0.39
NR1H4 Q96RI1 5/20 0.38
LPAR1 Q92633 1/20 0.38
LPAR2 Q9HBW0 1/20 0.38
LPAR3 Q9UBY5 1/20 0.38
SMPD1 P17405 2/20 0.36
PDE4A P27815 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2336634 0.93 LPAR1 (0.43) ALDH1A1THRBLPAR1LPAR2LPAR3
SCHEMBL3702563 0.92 NR1H4 (0.46) ALOX5ALOX5APPPARDNR1H4LPAR1
SCHEMBL3714445 0.88 LPAR1 (0.38) ALDH1A1NPC1RAB9ALPAR1LPAR2
SCHEMBL2339543 0.87 LPAR1 (0.42) ALDH1A1NPC1RAB9ATHRBLPAR1
SCHEMBL3717698 0.86 P2RX3 (0.38) ALDH1A1PPARDESR1THRATHRB
SCHEMBL3707582 0.86 LPAR1 (0.39) ALDH1A1NPC1RAB9ALPAR1LPAR2
SCHEMBL3700510 0.85 LPAR1 (0.36) ALDH1A1NPC1RAB9APPARDPPARG
SCHEMBL3710883 0.85 NR1H4 (0.48) PPARDESR1THRATHRBVDR
SCHEMBL3700609 0.84 LPAR1 (0.46) ALDH1A1PPARDNR1H4LPAR1LPAR2
SCHEMBL3704465 0.84 TBXAS1 (0.36) ALDH1A1ALOX5ALOX5APRXRALPAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010077882-A2 ANTAGONISTS OF LYSOPHOSPHATIDIC ACID RECEPTORS AMIRA PHARMACEUTICALS, INC. (US) 2010-07-08 WO disclosed