SCHEMBL3722649

SCHEMBL3722649

CN(C)CCSc1[c]ccc(-c2ccnc(N)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.43
HTR1A P08908 2/20 0.43
HRH3 Q9Y5N1 2/20 0.41
KMO O15229 1/20 0.40
AURKA O14965 2/20 0.38
HSP90AA1 P07900 1/20 0.38
PRKACA P17612 1/20 0.38
ADORA2A P29274 1/20 0.38
PIM1 P11309 6/20 0.38
PIM3 Q86V86 5/20 0.38
PIM2 Q9P1W9 5/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
CHUK O15111 1/20 0.36
PDPK1 O15530 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3715554 0.77 PIM1 (0.46) HRH3KMOAURKAHSP90AA1PRKACA
SCHEMBL3719906 0.72 ROCK2 (0.45) HTR7HTR1AAURKAPIM1PIM3
SCHEMBL3720566 0.69 KMO (0.43) KMOAURKAHSP90AA1PRKACAADORA2A
SCHEMBL10533843 0.67 HTR7 (0.59) HTR7HTR1ADRD2HTR2A
SCHEMBL5225822 0.67 MEN1 (0.54) HRH3AURKAHSP90AA1PRKACAADORA2A
SCHEMBL3656028 0.67 ROCK2 (0.60) HRH3KMOAURKAHSP90AA1PRKACA
SCHEMBL4703487 0.66 MEN1 (0.53) HRH3AURKAHSP90AA1PRKACAADORA2A
SCHEMBL4704184 0.65 HSP90AA1 (0.53) HTR7KMOAURKAHSP90AA1PRKACA
SCHEMBL3713494 0.64 CDK2 (0.39) KMOAURKAHSP90AA1PRKACAADORA2A
SCHEMBL10918299 0.62 KMO (0.57) KMOAURKAHSP90AA1PRKACAADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed