SCHEMBL3713494

SCHEMBL3713494

CCN(CC)C(=O)COc1[c]ccc(-c2ccnc(N)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.39
AURKA O14965 2/20 0.39
CHUK O15111 1/20 0.39
PDPK1 O15530 1/20 0.39
RPS6KB1 P23443 1/20 0.39
KDR P35968 1/20 0.39
TGFBR1 P36897 1/20 0.39
SYK P43405 1/20 0.39
JAK3 P52333 1/20 0.39
ROCK1 Q13464 1/20 0.39
AURKB Q96GD4 1/20 0.39
MAP3K5 Q99683 1/20 0.39
CDC7 O00311 3/20 0.39
DBF4 Q9UBU7 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ROCK2 O75116 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3813838 0.77 SLC2A1 (0.43) ROCK1KDM4EGAATDP1NPC1
SCHEMBL3715554 0.77 PIM1 (0.46) CDK2AURKACHUKPDPK1RPS6KB1
SCHEMBL3720566 0.72 KMO (0.43) CDK2AURKACHUKPDPK1RPS6KB1
SCHEMBL3661420 0.69 CDK2 (0.44) CDK2AURKACHUKPDPK1RPS6KB1
SCHEMBL8749753 0.69 RAB9A (0.54) KDM4EGAATDP1NPC1RAB9A
SCHEMBL3661410 0.67 CDC7 (0.50) CDK2CDC7DBF4ROCK2MAP4K4
SCHEMBL3717171 0.65 ROCK2 (0.41) ROCK1ROCK2GSK3BPRKACA
SCHEMBL3722649 0.64 HTR7 (0.43) CDK2AURKACHUKPDPK1RPS6KB1
SCHEMBL25305396 0.64 CDC7 (0.50) AURKASYKCDC7DBF4KDM4E
SCHEMBL5564786 0.62 ROCK1 (0.63) AURKAROCK1KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed