SCHEMBL3720566

SCHEMBL3720566

CN(C)C(=O)c1[c]ccc(-c2ccnc(N)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.43
JAK2 O60674 3/20 0.41
HSP90AA1 P07900 2/20 0.41
AURKA O14965 2/20 0.41
PRKACA P17612 1/20 0.41
ADORA2A P29274 1/20 0.41
HSP90AB1 P08238 1/20 0.40
PTK2 Q05397 1/20 0.40
CAMKK2 Q96RR4 1/20 0.40
CDK2 P24941 4/20 0.40
CDC7 O00311 4/20 0.40
CCNE1 P24864 2/20 0.40
DBF4 Q9UBU7 1/20 0.40
ROCK2 O75116 3/20 0.40
GSK3B P49841 2/20 0.40
MAP4K4 O95819 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
IRAK4 Q9NWZ3 1/20 0.40
CHUK O15111 1/20 0.39
PDPK1 O15530 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3713494 0.72 CDK2 (0.39) KMOHSP90AA1AURKAPRKACAADORA2A
SCHEMBL3715554 0.70 PIM1 (0.46) KMOHSP90AA1AURKAPRKACAADORA2A
SCHEMBL3722649 0.69 HTR7 (0.43) KMOHSP90AA1AURKAPRKACAADORA2A
SCHEMBL3661420 0.67 CDK2 (0.44) KMOHSP90AA1AURKAPRKACAADORA2A
SCHEMBL27115833 0.66 KMO (0.59) KMOHSP90AA1AURKAPRKACAADORA2A
SCHEMBL5397036 0.65 MAPK1 (0.49) JAK2HSP90AA1AURKAPRKACAADORA2A
SCHEMBL4704184 0.65 HSP90AA1 (0.53) KMOHSP90AA1AURKAPRKACAADORA2A
SCHEMBL7574364 0.65 ALDH1A1 (0.46) KDM4EALDH1A1MAPT
SCHEMBL10918299 0.65 KMO (0.57) KMOJAK2HSP90AA1AURKAPRKACA
SCHEMBL7584139 0.65 HPGD (0.40) KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed