SCHEMBL3725762

SCHEMBL3725762

COC(=O)c1csc(-c2cc3cc(C)cc([N+](=O)[O-])c3[nH]2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 4/20 0.44
MAOA P21397 1/20 0.41
ACHE P22303 1/20 0.41
RAB9A P51151 3/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 3/20 0.38
NPC1 O15118 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
FBP1 P09467 2/20 0.34
GPR35 Q9HC97 1/20 0.33
DCTPP1 Q9H773 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3031102 0.90 RAB9A (0.53) XDHRAB9AGAAMAPTNPC1
SCHEMBL27809827 0.88 ALDH1A1 (0.43) XDHACHERAB9AGAAGRIN2D
SCHEMBL3025131 0.85 MAOA (0.46) XDHMAOAACHERAB9AGAA
SCHEMBL27809770 0.81 XDH (0.36) XDHRAB9AMAPTNPC1MEN1
SCHEMBL27964610 0.79 GRIN2D (0.38) XDHMAPTMEN1KMT2AGRIN2D
SCHEMBL27809771 0.79 KDM4E (0.40) GAAMAPTMEN1KMT2AGRIN2D
SCHEMBL1278010 0.75 XDH (0.65) XDHRAB9AGAAMAPTNPC1
SCHEMBL14481501 0.70 ACHE (0.57) MAOAACHERAB9AMAPTNPC1
SCHEMBL3419709 0.69 GRIN2D (0.39) XDHMAPTGRIN2DGRIN3BGRIN1
SCHEMBL14656020 0.69 ACHE (0.64) MAOAACHERAB9AGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101801965-B Indole compounds as inhibitors of cellular necrosis LG LIFE SCIENCES LTD 2014-07-30 CN disclosed
EP-2178869-A1 INDOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG Life Sciences Ltd. (KR) 2010-04-28 EP disclosed
WO-2009025477-A1 INDOLE COMPOUNDS AS AN INHIBITOR OF CELLULAR NECROSIS LG LIFE SCIENCES LTD. (KR) 2009-02-26 WO disclosed