SCHEMBL3761968

SCHEMBL3761968

Cn1c(CN2CCCC2)ccc1C(=O)NCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.49
HTR1A P08908 1/20 0.48
HTR7 P34969 1/20 0.48
ALDH1A1 P00352 3/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
BRD4 O60885 1/20 0.44
KCNK3 O14649 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3772602 0.88 NPC1 (0.53) TP53ALDH1A1KDM4EGAAHPGD
N-Benzylmethylamine SCHEMBL5556336 0.84 NCF1 (0.50) HTR1AHTR7KMT2AKDM4E
SCHEMBL5189076 0.80 HTR1A (0.45) HTR1AHTR7ALDH1A1KMT2AKDM4E
SCHEMBL3762994 0.77 NPC1 (0.51) TP53ALDH1A1KDM4ELMNARAB9A
SCHEMBL3763647 0.76 HDAC3 (0.50) KMT2AMEN1
SCHEMBL13684982 0.76 SRC (0.47) TP53ALDH1A1L3MBTL1HPGDRAB9A
SCHEMBL22145190 0.74 ALDH1A1 (0.76) HTR1AHTR7ALDH1A1KMT2AMEN1
SCHEMBL3762346 0.73 HRH3 (0.50) ALDH1A1KDM4EGAAHPGD
SCHEMBL3761869 0.72 GAA (0.50) ALDH1A1KMT2AMEN1KDM4EGAA
SCHEMBL22145587 0.69 SIGMAR1 (0.60) TP53ALDH1A1KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842812-B2 Substituted 5-aminomethy1-1H-pyrrole-2-carboxylic acid amides GRUENENTHAL GMBH (DE) 2010-11-30 US disclosed
US-20070135494-A1 Substituted 5-aminomethyl-1H-pyrrole-2-carboxylic acid amides GRUENENTHAL GMBH (DE) 2007-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135494-A1 Substituted 5-aminomethyl-1H-pyrrole-2-carboxylic acid amides AVPR2, GPR119, AVPR1B TP53 4718/4885HTR1A 749/4885HTR7 813/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.