SCHEMBL3785285

SCHEMBL3785285

N=C(N)Nc1ccc(CCc2ccc(NC(=N)N)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.45
NPC1 O15118 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
NOS1 P29475 1/20 0.43
RAB9A P51151 1/20 0.43
HIF1A Q16665 1/20 0.43
SPHK1 Q9NYA1 4/20 0.43
BLM P54132 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
F2 P00734 1/20 0.41
PRSS1 P07477 1/20 0.41
PRSS2 P07478 1/20 0.41
PRSS3 P35030 1/20 0.41
TMPRSS6 Q8IU80 1/20 0.41
ST14 Q9Y5Y6 1/20 0.41
HRH3 Q9Y5N1 1/20 0.40
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13017226 0.90 AOC3 (0.46) AOC3NPC1CYP3A4CYP2D6NOS1
SCHEMBL13785815 0.90 AOC3 (0.40) AOC3NPC1CYP3A4CYP2D6NOS1
SCHEMBL13911596 0.90 TAAR1 (0.48) NPC1CYP3A4CYP2D6NOS1RAB9A
SCHEMBL2492523 0.90 CA2 (0.45) AOC3NPC1CYP3A4CYP2D6NOS1
Hydrochloric Acid SCHEMBL538308 0.88 ADRA2A (0.45) AOC3NPC1CYP3A4CYP2D6NOS1
SCHEMBL12514072 0.88 AOC3 (0.44) AOC3NPC1RAB9AGRIN2DGRIN3B
SCHEMBL7523474 0.88 SPHK1 (0.39) AOC3NPC1CYP3A4CYP2D6NOS1
SCHEMBL1743186 0.86 ADRA2A (0.50) F2PRSS1PRSS2PRSS3TMPRSS6
SCHEMBL1996992 0.85 F2 (0.50) NPC1CYP3A4CYP2D6RAB9AF2
SCHEMBL5447804 0.85 POLB (0.57) NPC1RAB9ASPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100331384-A1 GUANIDINE BASED COMPOUNDS UNIVERSIDAD DEL PAIS VASCO/EUSKAL HERRIKO UNIBERTSITATEA (ES) 2010-12-30 US disclosed
US-20100331384-A1 GUANIDINE BASED COMPOUNDS UNIVERSIDAD DEL PAIS VASCO/EUSKAL HERRIKO UNIBERTSITATEA (ES) 2010-12-30 US disclosed
US-20100331384-A1 GUANIDINE BASED COMPOUNDS UNIVERSIDAD DEL PAIS VASCO/EUSKAL HERRIKO UNIBERTSITATEA (ES) 2010-12-30 US disclosed
WO-2009080818-A2 GUANIDINE BASED COMPOUNDS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2009-07-02 WO disclosed
WO-2009080818-A2 GUANIDINE BASED COMPOUNDS THE PROVOST, FELLOWS AND SCHOLARS OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH NEAR DUBLIN (IE) 2009-07-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331384-A1 GUANIDINE BASED COMPOUNDS ADRB2, ADRA2A, ADRA2C AOC3 2450/4885NPC1 3544/4885CYP3A4 1380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.