Maleic Acid

Maleic Acid

SCHEMBL3797445

CCCCNCCCC.CCON1C(C)(C)CC(OC(C)=O)CC1(C)C.O=C(O)/C=C\C(=O)O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
TSHR P16473 2/20 0.41
ALDH1A1 P00352 1/20 0.37
ESR1 P03372 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
HCAR2 Q8TDS4 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL3797452 1.00 KMT2A (0.41) KMT2ATSHRALDH1A1ESR1HSD17B10
Fumaric Acid SCHEMBL3796830 0.90 TSHR (0.48) KMT2ATSHRALDH1A1ESR1HSD17B10
Maleic Acid SCHEMBL3796821 0.90 TSHR (0.48) KMT2ATSHRALDH1A1ESR1HSD17B10
Fumaric Acid SCHEMBL3796831 0.90 TSHR (0.48) KMT2ATSHRALDH1A1ESR1HSD17B10
SCHEMBL20073661 0.82 TSHR (0.51) KMT2ATSHRALDH1A1ESR1HSD17B10
SCHEMBL3797450 0.76 HCAR2 (0.33) HCAR2
SCHEMBL13130571 0.75 TSHR (0.39) KMT2ATSHRALDH1A1ESR1HSD17B10
SCHEMBL14706863 0.75 TSHR (0.45) KMT2ATSHRALDH1A1ESR1HSD17B10
SCHEMBL15850409 0.75 TSHR (0.45) KMT2ATSHRALDH1A1ESR1HSD17B10
SCHEMBL25699072 0.70 KMT2A (0.41) KMT2ATSHRALDH1A1ESR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8216596-B2 4-Hydroxy-1-(2-hydroxy-2-methylpropoxy)-2,2,6,6-tetramethylpiperidine, citric acid and a body care product; hindered amine salt compounds provide outstanding protection against light-induced fading BASF SE (DE) 2012-07-10 US claimed
EP-1893169-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CONTAINING STERICALLY HINDERED AMINE SALT COMPOUND Ciba Specialty Chemicals Holding Inc. (CH) 2008-03-05 EP claimed
US-20060262149-A1 Ink jet ink and recording material WOOD MERVIN G 2006-11-23 US claimed
US-20060264345-A1 Stabilized body care products, household products, textiles and fabrics BASF SE (DE) 2006-11-23 US claimed
WO-2006122888-A1 INK JET INK AND RECORDING MATERIAL CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-11-23 WO claimed
WO-2006122889-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CONTAINING STERICALLY HINDERED AMINE SALT COMPOUNDS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-11-23 WO claimed
US-8216596-B2 4-Hydroxy-1-(2-hydroxy-2-methylpropoxy)-2,2,6,6-tetramethylpiperidine, citric acid and a body care product; hindered amine salt compounds provide outstanding protection against light-induced fading BASF SE (DE) 2012-07-10 US disclosed
EP-2207522-A2 BODY-CARE AND HOUSEHOLD PRODUCTS AND COMPOSITIONS COMPRISING SPECIFIC SULFUR-CONTAINING COMPOUNDS BASF SE (DE) 2010-07-21 EP disclosed
WO-2009047150-A2 BODY-CARE AND HOUSEHOLD PRODUCTS AND COMPOSITIONS COMPRISING SPECIFIC SULFUR-CONTAINING COMPOUNDS BASF SE (CH) 2009-04-16 WO disclosed
US-20090092561-A1 Body-care and household products and compositions comprising specific sulfur-containing compounds BASF SE (DE) 2009-04-09 US disclosed
EP-1893169-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CONTAINING STERICALLY HINDERED AMINE SALT COMPOUND Ciba Specialty Chemicals Holding Inc. (CH) 2008-03-05 EP disclosed
US-20060262149-A1 Ink jet ink and recording material WOOD MERVIN G 2006-11-23 US disclosed
WO-2006122889-A2 STABILIZED BODY CARE PRODUCTS, HOUSEHOLD PRODUCTS, TEXTILES AND FABRICS CONTAINING STERICALLY HINDERED AMINE SALT COMPOUNDS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-11-23 WO disclosed
WO-2006122888-A1 INK JET INK AND RECORDING MATERIAL CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-11-23 WO disclosed
US-20060264345-A1 Stabilized body care products, household products, textiles and fabrics BASF SE (DE) 2006-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060264345-A1 Stabilized body care products, household products, textiles and fabrics DSC1, CUTA, DSG1 KMT2A 1031/4885TSHR 1283/4885ALDH1A1 1194/4885
US-20090092561-A1 Body-care and household products and compositions comprising specific sulfur-containing compounds DSC1, SCLY, DSG1 KMT2A 1820/4885TSHR 2447/4885ALDH1A1 1171/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.