SCHEMBL382838

SCHEMBL382838

CCOC(=O)c1ccc(N2CCC(NC3=NCCN3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 1/20 0.53
ITGB3 P05106 3/20 0.49
ITGAV P06756 3/20 0.49
ITGA2B P08514 3/20 0.49
ALDH1A1 P00352 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HSP90AA1 P07900 1/20 0.43
MAPT P10636 1/20 0.43
ADRA2A P08913 2/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
TSHR P16473 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
SIRT2 Q8IXJ6 2/20 0.41
SIRT1 Q96EB6 2/20 0.41
NOS2 P35228 1/20 0.40
METAP1 P53582 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382698 0.93 ITGB3 (0.53) PTGIRITGB3ITGAVITGA2BALDH1A1
SCHEMBL382510 0.81 NOS2 (0.51) ALDH1A1MEN1KMT2AHSP90AA1MAPT
SCHEMBL378108 0.76 MEN1 (0.50) ALDH1A1MEN1KMT2AHSP90AA1MAPT
Hydrochloric Acid SCHEMBL2514818 0.76 MEN1 (0.50) ALDH1A1MEN1KMT2AHSP90AA1TSHR
SCHEMBL384016 0.76 ITGB3 (0.56) ITGB3ITGAVITGA2BADRA2AADRA2B
SCHEMBL384017 0.76 ITGB3 (0.56) ITGB3ITGAVITGA2BADRA2AADRA2B
SCHEMBL8207095 0.75 HTT (0.52) ALDH1A1MEN1KMT2AHSP90AA1MAPT
SCHEMBL383015 0.74 OPRK1 (0.51) ALDH1A1MEN1KMT2AHSP90AA1MAPT
SCHEMBL382149 0.74 OPRK1 (0.51) ALDH1A1MEN1KMT2AHSP90AA1MAPT
SCHEMBL378276 0.74 TDP1 (0.60) ALDH1A1MEN1KMT2AHSP90AA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1074543-B1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA PHARMA CO LTD (JP) 2012-01-25 EP disclosed
US-6420558-B1 COMPOUNDS WITH AMIDINE GROUPS ANTAGONISTIC ACTIVITY, CELL ADHESION INHIBITORY ACTIVITY, HUMAN PLATELET AGGREGATION INHIBITORY ACTIVITY, AND THERAPEUTIC AGENTS MEIJI SEIKA KAISHA, LTD. (JP) 2002-07-16 US disclosed
EP-1074543-A1 AMINOPIPERIDINE DERIVATIVES AS INTEGRIN ALPHA V BETA 3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2001-02-07 EP disclosed