SCHEMBL3828659

SCHEMBL3828659

NS(=O)(=O)c1ccccc1-c1ccon1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 8/20 0.41
CA1 P00915 6/20 0.41
CA9 Q16790 5/20 0.41
CA6 P23280 3/20 0.41
CA12 O43570 3/20 0.41
CA4 P22748 2/20 0.41
CA5A P35218 2/20 0.41
CA7 P43166 2/20 0.41
CA5B Q9Y2D0 2/20 0.41
CYP2C9 P11712 1/20 0.41
CA14 Q9ULX7 1/20 0.41
ALOX5AP P20292 5/20 0.40
FEN1 P39748 5/20 0.40
STAT3 P40763 1/20 0.37
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27491067 0.79 CA2 (0.34) CA2CA1CA9CA6CA12
SCHEMBL28869430 0.79 NPC1 (0.41) CA2CA1CA9CA12CA4
SCHEMBL27536398 0.78 BRD4 (0.31)
SCHEMBL4059082 0.77 MDM2 (0.41) CYP2C9
SCHEMBL23235485 0.76 MDM2 (0.38) CA2CA1CA9STAT3
SCHEMBL10550462 0.75 ALOX5AP (0.43) CA2CA1CA9CA6CA12
SCHEMBL1080972 0.74 CA2 (0.61) CA2CA1CA9CA6CA12
Thiophene SCHEMBL27619739 0.72 CA1 (0.38) CA2CA1CA9CA12CA4
SCHEMBL8347239 0.72 CA2 (0.58) CA2CA1CA9CA6CA12
SCHEMBL8890179 0.72 PTPRC (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 206 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110521729-A A kind of composition pesticide and its application HEBEI ZHONGTIANBANGZHENG BIOLOGIC SCIENCE CO LTD 2019-12-03 CN claimed
CN-105358132-B Abuse resistant capsules R.P.谢勒技术有限公司 2019-10-15 CN claimed
CN-107232207-A A kind of herbicidal composition containing ring sulphur ketone, Garagard and isoxadifen 河南传奇农业科技有限公司 2017-10-10 CN claimed
CN-106818826-A A kind of crop phytocide composition 安徽常泰化工有限公司 2017-06-13 CN claimed
CN-103633062-B Compound semiconductor integrated circuit 稳懋半导体股份有限公司 2016-11-02 CN claimed
US-20030069287-A1 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors PHARMACIA CORPORATION 2003-04-10 US claimed
EP-1288206-A1 Substituted benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors G.D. SEARLE & CO. (US) 2003-03-05 EP claimed
US-6436967-B1 PREFERENTIAL CYCLOOXYGENASE INHIBITORS USED AS INJECTABLE ANALGESIC AND ANTIINFLAMMATORY AGENTS HAVING REDUCED SIDE EFFECTS; ACYLATION PHARMACIA CORPORATION 2002-08-20 US claimed
CN-106689202-B A kind of bactericidal composition 江苏龙灯化学有限公司 2019-11-22 CN disclosed
CN-209656599-U A kind of flash detecting device SHENZHEN FURUIKANG TECH CO LTD 2019-11-19 CN disclosed
CN-209656600-U A kind of flash detecting device SHENZHEN FURUIKANG TECH CO LTD 2019-11-19 CN disclosed
CN-209656598-U A kind of flash detecting device and X-ray excited polycrystalline structure scintillator SHENZHEN FURUIKANG TECH CO LTD 2019-11-19 CN disclosed
CN-209570532-U A kind of objective table driving assembly and detection device SHENZHEN FURUIKANG TECH CO LTD 2019-11-01 CN disclosed
CN-209570534-U A kind of darkroom component and detection device SHENZHEN FURUIKANG TECH CO LTD 2019-11-01 CN disclosed
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed
EP-0870764-A1 Sulfonamides and derivatives thereof that modulate the activity of endothelin TEXAS BIOTECHNOLOGY CORPORATION (US) 1998-10-14 EP disclosed
CN-1175411-A Use of dicafeoyl quininic acid in treatment of hepatitis B and diseases associated with retrovirus and cafeoyl quininic acid derivs. RADIOLOGY INST MILITARY MEDICA (CN) 1998-03-11 CN disclosed
US-5571821-A CARDIOVASCULAR DISORDERS TO MODULATE ENDOTHELIN, HYPOTENSIVE AGENTS AND VASOCONSTRICTION TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-11-05 US disclosed
EP-0699191-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN TEXAS BIOTECHNOLOGY CORPORATION (US) 1996-03-06 EP disclosed
WO-1994027979-A1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN IMMUNOPHARMACEUTICS, INC. (US) 1994-12-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030069287-A1 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors PTGS2, PTGES2, PTGES CA2 920/4885CA1 2057/4885CA9 1174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.