SCHEMBL38428

SCHEMBL38428

CCOC(=O)N1CCC(NC(=O)NCc2cccc(-c3cn4ncccc4n3)c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.46
KDM4E B2RXH2 8/20 0.46
MAPT P10636 3/20 0.46
NPC1 O15118 1/20 0.46
ATM Q13315 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
HPGD P15428 5/20 0.45
HSD17B10 Q99714 4/20 0.45
ALOX15 P16050 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
LMNA P02545 1/20 0.45
EPHX2 P34913 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MAPK1 P28482 2/20 0.42
USP2 O75604 1/20 0.42
NOS2 P35228 1/20 0.41
WDR5 P61964 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44576 0.76 WDR5 (0.46) ALDH1A1KDM4EMAPTSMN1; SMN2WDR5
SCHEMBL38703 0.75 WDR5 (0.44) ALDH1A1KDM4EHPGDWDR5
SCHEMBL39537 0.74 WDR5 (0.46) ALDH1A1KDM4EMAPTHPGDHSD17B10
SCHEMBL38565 0.74 WDR5 (0.44) ALDH1A1KDM4ENPC1ATMHPGD
SCHEMBL39240 0.72 BTK (0.43) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL44622 0.72 LMNA (0.50) ALDH1A1KDM4EMAPTNPC1MEN1
SCHEMBL44301 0.71 WDR5 (0.66) ALDH1A1KDM4ENPC1HPGDHSD17B10
SCHEMBL38716 0.71 FBP1 (0.47) ALDH1A1KDM4EMAPTSMN1; SMN2WDR5
SCHEMBL44216 0.71 WDR5 (0.52) NPC1HPGDLMNAWDR5
SCHEMBL44512 0.69 WDR5 (0.52) KDM4EMAPTNPC1LMNAWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed