SCHEMBL389392

SCHEMBL389392

O/C(=C/c1ccccc1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.54
MAPT P10636 3/20 0.52
MEN1 O00255 2/20 0.52
HTT P42858 2/20 0.52
KMT2A Q03164 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
PRMT1 Q99873 1/20 0.48
ESR1 P03372 1/20 0.48
CYP19A1 P11511 4/20 0.46
CYP11B2 P19099 2/20 0.46
NFE2L2 Q16236 1/20 0.46
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
KDM4E B2RXH2 1/20 0.45
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL918848 1.00 AKR1C1 (0.54) AKR1C1MAPTMEN1HTTKMT2A
SCHEMBL368124 1.00 AKR1C1 (0.54) AKR1C1MAPTMEN1HTTKMT2A
SCHEMBL9950184 0.85 ESR1 (0.57) MAPTMEN1HTTKMT2ANPC1
Cinnamic Acid SCHEMBL17240386 0.82 HCAR2 (0.70) AKR1C1MAPTMEN1KMT2ARAB9A
SCHEMBL2495017 0.80 KMO (0.52) AKR1C1PRMT1
SCHEMBL22829697 0.80 CHAT (0.55) AKR1C1MAPTMEN1HTTKMT2A
SCHEMBL14836770 0.79 AKR1C1 (0.56) AKR1C1MAPTMEN1HTTKMT2A
SCHEMBL19433105 0.79 PTGS1 (0.47) MAPTMEN1HTTKMT2ANPC1
SCHEMBL9858496 0.79 MAPT (0.58) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL1647472 0.78 ALDH1A1 (0.44) AKR1C1MEN1KMT2APRMT1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1845957-B1 METHOD FOR PRODUCING A DRUG EXTRACT THAT CONTAINS HYDROXYSTILBENES HEGER PETER (DE) 2010-12-22 EP claimed
WO-2010049390-A1 COSMETIC AND DERMATOLOGICAL COMPOSITIONS FOR THE REDUCTION OF FACIAL EXPRESSION WRINKLES HENKEL AG & CO. KGAA (DE) 2010-05-06 WO claimed
EP-1844784-B1 A pharmaceutical composition for the treatment of pathologies caused by the general response of the immune system EPITECH GROUP SRL (IT) 2010-04-21 EP claimed
EP-2005941-A2 Cellular rejuvenation compounds Henkel AG & Co. KGaA (DE) 2008-12-24 EP claimed
EP-1845957-A1 METHOD FOR PRODUCING A DRUG EXTRACT THAT CONTAINS HYDROXYSTILBENE Heger, Peter (DE) 2007-10-24 EP claimed
WO-2006082071-A1 METHOD FOR PRODUCING A DRUG EXTRACT THAT CONTAINS HYDROXYSTILBENE HEGER PETER (DE) 2006-08-10 WO claimed
EP-2238968-B1 Skin treatment fighting skin aging HENKEL AG & CO KGAA (DE) 2018-05-02 EP disclosed
EP-2238967-B1 Skin treatment fighting skin aging II HENKEL AG & CO KGAA (DE) 2018-05-02 EP disclosed
EP-2202215-B1 Novel process for the synthesis of (E)-Stilbene derivatives which makes it possible to obtain resveratrol and piceatannol CLARIANT SPECIALTY FINE CHEM F (FR) 2013-10-02 EP disclosed
EP-2049459-B1 NOVEL PROCESS FOR THE SYNTHESIS OF (E)-STILBENE DERIVATIVES WHICH MAKES IT POSSIBLE TO OBTAIN RESVERATROL AND PICEATANNOL CLARIANT SPECIALTY FINE CHEM F (FR) 2013-10-02 EP disclosed
US-8101804-B2 Process for the synthesis of (E)-stilbene derivatives which makes it possible to obtain resveratrol and piceatannol CLARIANT SPECIALTY FINE CHEMICALS (FRANCE) (FR) 2012-01-24 US disclosed
EP-2238967-A2 Skin treatment fighting skin aging II Henkel AG & Co. KGaA (DE) 2010-10-13 EP disclosed
EP-2238968-A2 Skin treatment fighting skin aging Henkel AG & Co. KGaA (DE) 2010-10-13 EP disclosed
US-20080119649-A1 HALOCOMBSTATINS AND METHODS OF SYNTHESIS THEREOF ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA, ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY 2008-05-22 US disclosed
WO-2008012321-A1 NOVEL PROCESS FOR THE SYNTHESIS OF (E)-STILBENE DERIVATIVES WHICH MAKES IT POSSIBLE TO OBTAIN RESVERATROL AND PICEATANNOL CLARIANT SPECIALTY FINE CHEMICALS (FRANCE) (FR) 2008-01-31 WO disclosed
US-20070167412-A1 HALOCOMBSTATINS AND METHODS OF SYNTHESIS THEREOF ARIZONA BOARD OF REGENTS (US) 2007-07-19 US disclosed
EP-1802560-A2 HALOCOMBSTATINS AND METHODS OF SYNTHESIS THEREOF Arizona Board Regents, a body corporate of the State of Arizona, acting for and on behalf of Arizona State University (US) 2007-07-04 EP disclosed
US-7223747-B2 Halocombstatins and methods of synthesis thereof ARIZONA BOARD OF REGENTS ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2007-05-29 US disclosed
WO-2006036743-A2 HALOCOMBSTATINS AND METHODS OF SYNTHESIS THEREOF ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2006-04-06 WO disclosed
US-20050176688-A1 Halocombstatins and methods of synthesis thereof ARIZONA BOARD OF REGENTS, A BODY CORPORATE OF THE STATE OF ARIZONA 2005-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080119649-A1 HALOCOMBSTATINS AND METHODS OF SYNTHESIS THEREOF TUBB3, TUBB8B, TUBB8 AKR1C1 3954/4885MAPT 258/4885MEN1 2337/4885
US-20070167412-A1 HALOCOMBSTATINS AND METHODS OF SYNTHESIS THEREOF TUBB3, TUBB8B, TUBB8 AKR1C1 3954/4885MAPT 258/4885MEN1 2337/4885
US-20050176688-A1 Halocombstatins and methods of synthesis thereof TUBB3, TUBB8B, TUBB8 AKR1C1 3954/4885MAPT 258/4885MEN1 2337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.