SCHEMBL3900527

SCHEMBL3900527

CN(C)C(=O)c1ccc(C(N)=O)c(CCOc2cc(C#N)ccc2I)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.36
PDK1 Q15118 2/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
CDK8 P49336 2/20 0.36
CCNC P24863 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
F10 P00742 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 2/20 0.33
KCNH2 Q12809 2/20 0.32
KDR P35968 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3900535 0.76 NPC1 (0.43) CDK1ALDH1A1EGLN1
SCHEMBL3900423 0.67 F10 (0.43) CDK1PDK1PDK2PDK3PDK4
SCHEMBL28223333 0.67 KDR (0.41) ALDH1A1KCNH2KDRPIK3CAPIK3CB
SCHEMBL3905446 0.67 KDM4E (0.40) CYP11B1CYP11B2TTRPARP2PTGDR2
SCHEMBL3900652 0.66 RAB9A (0.46) CDK1F10EGLN1
SCHEMBL9850808 0.66 MAPT (0.47) ALDH1A1MAPTSLC6A3KCNH2KDR
Hydrochloric Acid SCHEMBL3896102 0.65 KDM4E (0.43) CYP11B1CYP11B2ALDH1A1PARP2PTGDR2
SCHEMBL24022839 0.65 CASP1 (0.44) KCNH2KDRPIK3CAPIK3CBMTOR
SCHEMBL3896082 0.65 MMP3 (0.44) CYP11B1CYP11B2TTREGLN1PTGDR2
SCHEMBL3571548 0.64 TRPV4 (0.40) MAPTSLC6A4KCNH2TTRPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0976722-B1 BENZAMIDINE DERIVATIVES AJINOMOTO KK (JP) 2009-03-11 EP disclosed
US-7396844-B1 Benzamidine derivatives AJINOMOTO CO., INC. (JP) 2008-07-08 US disclosed
EP-0976722-A1 BENZAMIDINE DERIVATIVES Ajinomoto Co., Inc. (JP) 2000-02-02 EP disclosed