Diamide

Diamide

SCHEMBL3943566

CCOC(C)OCC.CN(C)C(=O)N=NC(=O)N(C)C

nearest known ligand 0.54

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
TSHR P16473 1/20 0.54
NFKB1 P19838 1/20 0.54
THPO P40225 1/20 0.54
HSD17B10 Q99714 1/20 0.54
MAPT P10636 1/20 0.54
APEX1 P27695 1/20 0.54
PMP22 Q01453 1/20 0.54
LMNA P02545 1/20 0.50
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5907461 0.80 LMNA (0.57) ALDH1A1HSD17B10MAPTLMNACHRNB2
Diamide SCHEMBL5320404 0.78 ALDH1A1 (0.65) ALDH1A1TSHRNFKB1THPOHSD17B10
Butane SCHEMBL3151311 0.77 LMNA (0.52) ALDH1A1HSD17B10LMNACHRNB2CHRNB4
Butane SCHEMBL3150354 0.75 LMNA (0.50) ALDH1A1LMNACHRNB2CHRNB4CHRNA4
Butane SCHEMBL10560420 0.75 LMNA (0.44) ALDH1A1LMNACHRNB2CHRNB4CHRNA4
Bicarbonate SCHEMBL5374586 0.74 LMNA (0.71) ALDH1A1HSD17B10LMNA
Bicarbonate SCHEMBL28895866 0.74 LMNA (0.71) ALDH1A1HSD17B10LMNA
Acetone SCHEMBL590699 0.74 LMNA (0.71) ALDH1A1TSHRHSD17B10LMNA
Bicarbonate SCHEMBL28942687 0.74 LMNA (0.71) ALDH1A1HSD17B10LMNA
Diamide SCHEMBL1302348 0.74 ALDH1A1 (0.77) ALDH1A1TSHRNFKB1THPOHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794205-B1 METHACRYLATE AMIDE ACETALS IN COATINGS DU PONT (US) 2012-06-13 EP disclosed
US-7608645-B2 Use of (meth)acrylate functionalized amide acetals as reactive components with crosslinking agents and UV radiation; coating can be crosslinked by reaction with a crosslinker, such as isocyanate, and subsequently cured additionally by exposure to UV or electron beam (EB) energy; hardness, clarity E.I. DU PONT DE NEMOURS AND COMPANY (US) 2009-10-27 US disclosed
EP-1794166-B1 POLYMERIC/OLIGOMERIC METHACRYLATE FUNCTIONALIZED AMIDE ACETALS IN COATINGS DU PONT (US) 2009-08-19 EP disclosed
US-7504459-B2 Methacrylate amide acetals in coatings E.I. DU PONT DE NEMOURS & COMPANY (US) 2009-03-17 US disclosed
EP-1670840-B1 PROCESS FOR MAKING AMIDE ACETALS DU PONT (US) 2008-09-03 EP disclosed
EP-1805185-A1 HYDROXY AMIDE ACETALS AND THEIR USE IN COATINGS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2007-07-11 EP disclosed
EP-1794166-A1 POLYMERIC/OLIGOMERIC METHACRYLATE FUNCTIONALIZED AMIDE ACETALS IN COATINGS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2007-06-13 EP disclosed
EP-1794205-A1 METHACRYLATE AMIDE ACETALS IN COATINGS E.I. du Pont de Nemours & Company (US) 2007-06-13 EP disclosed
US-7230112-B2 Process for making amide acetals E. I. DUPONT DE NEMOURS AND COMPANY (US) 2007-06-12 US disclosed
US-7135530-B2 Polymeric/oligomeric methacrylate functionalized amide acetals in coatings E. I. DU PONT DE NEMOURS AND COMPANY (US) 2006-11-14 US disclosed
EP-1670840-A1 PROCESS FOR MAKING AMIDE ACETALS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2006-06-21 EP disclosed
US-20060128873-A1 Dual cure coating compositions AXALTA COATING SYSTEMS IP CO. LLC (FORMERLY KNOWN AS U.S. COATINGS IP CO. LLC) 2006-06-15 US disclosed
WO-2006039618-A1 POLYMERIC/OLIGOMERIC METHACRYLATE FUNCTIONALIZED AMIDE ACETALS IN COATINGS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2006-04-13 WO disclosed
WO-2006039619-A1 HYDROXY AMIDE ACETALS AND THEIR USE IN COATINGS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2006-04-13 WO disclosed
WO-2006039617-A1 METHACRYLATE AMIDE ACETALS IN COATINGS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2006-04-13 WO disclosed
US-20060069233-A1 Polymeric/oligomeric methacrylate functionalized amide acetals in coatings AXALTA COATING SYSTEMS IP CO. LLC (FORMERLY KNOWN AS U.S. COATINGS IP CO. LLC) 2006-03-30 US disclosed
US-20060069205-A1 Hydroxy amide acetals in coatings E. I. DU PONT DE NEMOURS AND COMPANY 2006-03-30 US disclosed
US-20060069204-A1 Methacrylate amide acetals in coatings AXALTA COATING SYSTEMS IP CO. LLC (FORMERLY KNOWN AS U.S. COATINGS IP CO. LLC) 2006-03-30 US disclosed
US-20050222425-A1 Process for making amide acetals AXALTA COATING SYSTEMS IP CO. LLC (FORMERLY KNOWN AS U.S. COATINGS IP CO. LLC) 2005-10-06 US disclosed
WO-2005035613-A1 PROCESS FOR MAKING AMIDE ACETALS E.I. DUPONT DE NEMOURS AND COMPANY (US) 2005-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050222425-A1 Process for making amide acetals NAAA, APEH, AMDHD2 ALDH1A1 213/4885TSHR 4463/4885NFKB1 2536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.