Cariporide

Cariporide

SCHEMBL39639

CC(C)c1ccc(C(=O)NC(=N)N)cc1S(C)(=O)=O

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 3/20 0.61
SLC9A2 Q9UBY0 1/20 0.60
CNR2 P34972 1/20 0.41
PLAU P00749 1/20 0.38
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
SCN5A Q14524 2/20 0.36
SCN2A Q99250 2/20 0.36
F10 P00742 2/20 0.34
PRSS1 P07477 2/20 0.34
PRSS2 P07478 2/20 0.34
PRSS3 P35030 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cariporide SCHEMBL6261845 0.99 SLC9A1 (0.63) SLC9A1SLC9A2CNR2PLAUCA1
Cariporide SCHEMBL221094 0.99 SLC9A1 (0.63) SLC9A1SLC9A2CNR2PLAUCA1
Cariporide SCHEMBL1229789 0.99 SLC9A1 (0.60) SLC9A1SLC9A2CNR2PLAUCA1
Cariporide SCHEMBL220085 0.99 SLC9A1 (0.60) SLC9A1SLC9A2CNR2PLAUCA1
Hydrochloric Acid SCHEMBL8816752 0.88 SLC9A1 (0.47) SLC9A1SLC9A2CNR2PLAUCA1
SCHEMBL8743805 0.87 SLC9A1 (0.47) SLC9A1SLC9A2PLAUCA1CA2
Hydrochloric Acid SCHEMBL8743814 0.86 SLC9A1 (0.46) SLC9A1SLC9A2PLAUCA1CA2
Hydrochloric Acid SCHEMBL8983516 0.86 SLC9A1 (0.46) SLC9A1SLC9A2PLAUCA1CA2
SCHEMBL8647598 0.85 SLC9A1 (0.44) SLC9A1SLC9A2CNR2PLAUCA1
Cariporide SCHEMBL936191 0.84 ALDH1A1 (0.48) SLC9A1SLC9A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1739 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260053134-A1 PERFUSION SOLUTION ORGAN TRANSP PTY LTD (AU) 2026-02-26 US claimed
EP-4577202-A1 USE OF A THERAPEUTIC AGENT WITH SODIUM-HYDROGEN ANTIPORTER 1 INHIBITORY ACTIVITY FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERTIONAL INTOLERANCE Mitodicure GmbH (DE) 2025-07-02 EP claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
US-20250049747-A1 USE OF HYPERPOLARIZING AGENTS ALONE AND IN COMBINATION WITH OTHER THERAPEUTIC AGENTS FOR TREATING CANCERS INCLUDING GLIOBLASTOMA TRUSTEES OF TUFTS COLLEGE 2025-02-13 US claimed
EP-4447955-A1 USE OF HYPERPOLARIZING AGENTS ALONE AND IN COMBINATION WITH OTHER THERAPEUTIC AGENTS FOR TREATING CANCERS INCLUDING GLIOBLASTOMA Trustees of Tufts College (US) 2024-10-23 EP claimed
US-20240334925-A9 PERFUSION SOLUTION PERFUSION FLUID TECHNOLOGIES INC (US) 2024-10-10 US claimed
US-12082575-B2 Perfusion solution Organ Transport Pty Ltd (AU) 2024-09-10 US claimed
US-20240090494-A1 PERFUSION SOLUTION ORGAN TRANSP PTY LTD (AU) 2024-03-21 US claimed
WO-2024042160-A1 USE OF A THERAPEUTIC AGENT WITH SODIUM-HYDROGEN ANTIPORTER 1 INHIBITORY ACTIVITY FOR THE TREATMENT AND PREVENTION OF DISEASES ASSOCIATED WITH CHRONIC FATIGUE, EXHAUSTION AND/OR EXERTIONAL INTOLERANCE MITODICURE GMBH (DE) 2024-02-29 WO claimed
US-20240041804-A1 NHE-1 INHIBITORS FOR THE TREATMENT OF CORONAVIRUS INFECTIONS FONDATION ESPERARE (CH) 2024-02-08 US claimed
WO-2001045716-A1 PHARMACEUTICAL COMPOSITION COMPRISING A PHYSIOLOGICALLY ACCEPTABLE VANADIUM COMPOUND, SALT OR COMPLEX AND A NA+/H+ EXCHANGE INHIBITOR GHO'ST HOLDING B.V. (NL) 2001-06-28 WO claimed
WO-2000067756-A1 METHODS FOR CONTROLLING INTRAOCULAR PRESSURE THE TRUSTEES OF THE UNIVERSTIY OF PENNSYLVANIA (US) 2000-11-16 WO claimed
WO-2000038661-A2 THE UTILISATION OF INHIBITORS OF THE SODIUM HYDROGEN EXCHANGER FOR PRODUCING A MEDICAMENT FOR PREVENTING ORGAN DYSFUNCTIONS AND DISEASES RELATED TO A PARTICULAR AGE AND FOR PROLONGING LIFE AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-07-06 WO claimed
EP-0950418-A2 Composition for preventing or treating ischemic disease Takeda Chemical Industries, Ltd. (JP) 1999-10-20 EP claimed
EP-0937464-A2 Combined pharmaceutical preparation containing inhibitors of the sodium hydrogen exchange and a medicament for the treatment of cardiovascular diseases Hoechst Marion Roussel Deutschland GmbH (DE) 1999-08-25 EP claimed
EP-0916337-A2 Use of inhibitors of the sodium-hydrogen exchange in the manufacture of amedicament for reducing unwanted effects of compounds on the heart. Hoechst Marion Roussel Deutschland GmbH (DE) 1999-05-19 EP claimed
EP-0909559-A2 Use of inhibitors of the sodium hydrogen exchange in the manufacture of a medicament for treatment or prophylaxis of diseases of the central nervous system Hoechst Marion Roussel Deutschland GmbH (DE) 1999-04-21 EP claimed
CN-1212149-A Use of inhibitor of Na+/H+ exchanger for production of medicament HOECHST MARION ROUSSEL DE GMBH (DE) 1999-03-31 CN claimed
CN-1209995-A Use of sodium-hydrogen exchanger inhibitors for the production of a medicament for reducing the adverse effects of substances on the heart HOECHST MARION ROUSSEL DE GMBH (DE) 1999-03-10 CN claimed
CN-1209316-A Combined medicinal preparation of sodium/hydrogen exchange-pump inhibitor and medicine for treatment of angiocardiopathy HOECHST MARION ROUSSEL DE GMBH (DE) 1999-03-03 CN claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240041804-A1 NHE-1 INHIBITORS FOR THE TREATMENT OF CORONAVIRUS INFECTIONS NHERF1, SLC9A1, SLC9A2 SLC9A1 2/4885SLC9A2 3/4885CNR2 1955/4885
US-20250049747-A1 USE OF HYPERPOLARIZING AGENTS ALONE AND IN COMBINATION WITH OTHER THERAPEUTIC AGENTS FOR TREATING CANCERS INCLUDING GLIOBLASTOMA MTOR, KCNN1, HCN4 SLC9A1 25/4885SLC9A2 27/4885CNR2 1274/4885
US-20260053134-A1 PERFUSION SOLUTION ATP2A1, SLC8B1, GLS SLC9A1 63/4885SLC9A2 155/4885CNR2 4095/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.