SCHEMBL39660

SCHEMBL39660

COc1ccc(S(=O)(=O)NCc2cccc(-c3cn4cc(C)sc4n3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.56
ALDH1A1 P00352 4/20 0.49
THRB P10828 1/20 0.48
RECQL P46063 1/20 0.48
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 3/20 0.44
LMNA P02545 2/20 0.44
TP53 P04637 1/20 0.44
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
TSHR P16473 1/20 0.43
AURKA O14965 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL39342 0.89 CYP19A1 (0.53) CYP19A1ALDH1A1KMT2AMEN1POLB
SCHEMBL44780 0.84 ALDH1A1 (0.44) CYP19A1ALDH1A1KMT2AMEN1MAPT
SCHEMBL44302 0.84 SMN1; SMN2 (0.50) CYP19A1ALDH1A1KMT2AMEN1POLB
SCHEMBL44636 0.82 TP53 (0.43) CYP19A1ALDH1A1THRBKMT2AMEN1
SCHEMBL44557 0.82 KMT2A (0.40) CYP19A1ALDH1A1THRBKMT2AMEN1
SCHEMBL44918 0.82 CYP19A1 (0.44) CYP19A1ALDH1A1POLBMAPTLMNA
SCHEMBL45229 0.80 TP53 (0.41) CYP19A1ALDH1A1THRBKMT2AMEN1
SCHEMBL44139 0.80 ALDH1A1 (0.43) CYP19A1ALDH1A1THRBMAPTLMNA
SCHEMBL44674 0.76 MAPT (0.52) POLBMAPTTP53
SCHEMBL44862 0.76 GAA (0.47) CYP19A1ALDH1A1THRBPOLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed