SCHEMBL45229

SCHEMBL45229

Cc1cn2cc(-c3cccc(CNS(=O)(=O)c4ccccc4F)c3)nc2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.41
NR3C2 P08235 2/20 0.40
NR3C1 P04150 1/20 0.39
POLB P06746 3/20 0.39
PKM P14618 1/20 0.38
CYP19A1 P11511 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
MAPT P10636 4/20 0.38
THRB P10828 1/20 0.38
KAT6A Q92794 2/20 0.37
PI4KB Q9UBF8 1/20 0.37
CNR1 P21554 1/20 0.37
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
LMNA P02545 3/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44557 0.90 KMT2A (0.40) TP53NR3C2POLBCYP19A1SMN1; SMN2
SCHEMBL44139 0.89 ALDH1A1 (0.43) TP53NR3C2CYP19A1SMN1; SMN2MAPT
SCHEMBL39342 0.86 CYP19A1 (0.53) TP53POLBCYP19A1SMN1; SMN2MAPT
SCHEMBL44302 0.85 SMN1; SMN2 (0.50) TP53POLBCYP19A1SMN1; SMN2MAPT
SCHEMBL44636 0.83 TP53 (0.43) TP53CYP19A1SMN1; SMN2MAPTTHRB
SCHEMBL44780 0.81 ALDH1A1 (0.44) TP53PKMCYP19A1SMN1; SMN2MAPT
SCHEMBL39660 0.80 CYP19A1 (0.56) TP53POLBCYP19A1MAPTTHRB
SCHEMBL44918 0.79 CYP19A1 (0.44) TP53NR3C2POLBCYP19A1SMN1; SMN2
SCHEMBL44862 0.77 GAA (0.47) TP53POLBCYP19A1SMN1; SMN2MAPT
SCHEMBL44054 0.76 MAPT (0.53) TP53SMN1; SMN2MAPTTHRBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed