SCHEMBL44918

SCHEMBL44918

Cc1cn2cc(-c3cccc(CNS(=O)(=O)c4cccc(C#N)c4)c3)nc2s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.44
NAMPT P43490 1/20 0.41
NR3C2 P08235 1/20 0.41
MAPT P10636 4/20 0.40
ALDH1A1 P00352 3/20 0.40
USP2 O75604 2/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HSD17B1 P14061 1/20 0.39
HSD17B2 P37059 1/20 0.39
SCN9A Q15858 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CG P48736 1/20 0.38
KDM4E B2RXH2 2/20 0.37
BRD4 O60885 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44780 0.86 ALDH1A1 (0.44) CYP19A1MAPTALDH1A1USP2LMNA
SCHEMBL44302 0.86 SMN1; SMN2 (0.50) CYP19A1NAMPTMAPTALDH1A1USP2
SCHEMBL44750 0.85 CYP1A2 (0.41) CYP19A1MAPTALDH1A1USP2LMNA
SCHEMBL39342 0.83 CYP19A1 (0.53) CYP19A1MAPTALDH1A1USP2LMNA
SCHEMBL39660 0.82 CYP19A1 (0.56) CYP19A1MAPTALDH1A1LMNAHSD17B1
SCHEMBL44636 0.81 TP53 (0.43) CYP19A1MAPTALDH1A1USP2LMNA
SCHEMBL44557 0.81 KMT2A (0.40) CYP19A1NR3C2MAPTALDH1A1USP2
SCHEMBL45229 0.79 TP53 (0.41) CYP19A1NR3C2MAPTALDH1A1USP2
SCHEMBL44139 0.79 ALDH1A1 (0.43) CYP19A1NR3C2MAPTALDH1A1USP2
SCHEMBL44398 0.78 CHRM3 (0.52) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed