SCHEMBL44139

SCHEMBL44139

Cc1cn2cc(-c3cccc(CNS(=O)(=O)c4ccccc4Cl)c3)nc2s1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 6/20 0.40
TP53 P04637 5/20 0.40
MAPT P10636 4/20 0.40
NR3C2 P08235 1/20 0.40
LMNA P02545 3/20 0.39
SLC12A2 P55011 1/20 0.39
SLC12A5 Q9H2X9 1/20 0.39
GLA P06280 1/20 0.39
HSD11B1 P28845 1/20 0.38
THRB P10828 2/20 0.38
HSD17B1 P14061 1/20 0.37
HSD17B2 P37059 1/20 0.37
USP2 O75604 2/20 0.36
HTT P42858 1/20 0.36
CYP19A1 P11511 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL44557 0.90 KMT2A (0.40) ALDH1A1SMN1; SMN2TP53MAPTNR3C2
SCHEMBL45229 0.89 TP53 (0.41) ALDH1A1SMN1; SMN2TP53MAPTNR3C2
SCHEMBL44780 0.85 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL44636 0.83 TP53 (0.43) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL39342 0.82 CYP19A1 (0.53) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL44302 0.81 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL39660 0.80 CYP19A1 (0.56) ALDH1A1TP53MAPTLMNATHRB
SCHEMBL44918 0.79 CYP19A1 (0.44) ALDH1A1SMN1; SMN2TP53MAPTNR3C2
SCHEMBL44862 0.77 GAA (0.47) ALDH1A1SMN1; SMN2TP53MAPTLMNA
SCHEMBL44400 0.76 ALDH1A1 (0.45) ALDH1A1TP53NR3C2LMNASLC12A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO claimed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed
WO-2011137587-A1 CYTOKINE INHIBITORS HUTCHISON MEDIPHARMA LIMITED (CN) 2011-11-10 WO disclosed