SCHEMBL3989519

SCHEMBL3989519

CC(C)C(NC(=O)C(Cc1ccc(F)cc1)NC(=O)OCc1ccccc1)C(=O)N(C)C(Cc1ccc(O)c(C(C)(C)C)c1)c1nnco1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.38
CASP7 P55210 1/20 0.38
REN P00797 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
OPRK1 P41145 1/20 0.37
CASP1 P29466 2/20 0.37
CASP9 P55211 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3988196 0.79 CA2 (0.42) CASP3CASP7MEN1KMT2ACASP1
SCHEMBL3989682 0.76 TACR1 (0.48) MEN1KMT2ACTSLCTSBCTSS
SCHEMBL3987520 0.73 CTSL (0.41) CASP3CASP7MEN1KMT2ACTSL
SCHEMBL8815629 0.72 CTSB (0.62) CASP3CASP7RENCTSLCTSB
SCHEMBL8815632 0.72 CTSB (0.62) CASP3CASP7RENCTSLCTSB
SCHEMBL5686625 0.71 CTSB (0.57) CASP3CASP7RENCTSLCTSB
SCHEMBL3989402 0.70
SCHEMBL7788731 0.69 CA4 (0.41) CASP3CASP7CTSLCTSBCTSS
SCHEMBL23447154 0.67 CTSS (0.54) RENCTSLCTSBCTSSCTSK
SCHEMBL3987548 0.67 ERCC1 (0.30) RENCTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed