SCHEMBL3989682

SCHEMBL3989682

CC(C)(C)c1cc(CC(NC(=O)OCc2ccccc2)c2nnco2)ccc1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.48
ATM Q13315 1/20 0.44
MAPT P10636 2/20 0.41
ALDH1A1 P00352 4/20 0.39
TSHR P16473 3/20 0.39
LMNA P02545 3/20 0.39
HPGD P15428 3/20 0.39
HTT P42858 3/20 0.39
NPSR1 Q6W5P4 3/20 0.39
PKM P14618 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TP53 P04637 1/20 0.39
AGTR1 P30556 1/20 0.39
RAB9A P51151 1/20 0.39
XBP1 P17861 2/20 0.39
MEN1 O00255 1/20 0.39
ALOX15 P16050 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CTSL P07711 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3988196 0.92 CA2 (0.42) TACR1ATMMEN1KMT2A
SCHEMBL27553310 0.84 TACR1 (0.47) TACR1ATMMAPTALDH1A1TSHR
SCHEMBL3995160 0.79 REN (0.33) ATMALDH1A1NPSR1XBP1CTSL
SCHEMBL3988336 0.78 PTPRB (0.46) TACR1ATMCTSLCTSBCTSS
SCHEMBL3987548 0.78 ERCC1 (0.30) CTSLCTSS
SCHEMBL3989464 0.78 CTSL (0.45) TACR1CTSLCTSBCTSSCTRB1
SCHEMBL3989460 0.78 CTSL (0.45) TACR1CTSLCTSBCTSSCTRB1
SCHEMBL17357789 0.77 ATM (0.52) TACR1ATMMAPTSMN1; SMN2CTSL
SCHEMBL3989467 0.77 CTSB (0.50) CTSLCTSBCTSSCTRB1SYK
SCHEMBL3989519 0.76 CASP3 (0.38) MEN1KMT2ACTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7553969-B1 Substituted phenethylamine derivatives CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-06-30 US disclosed
EP-1149843-A1 SUBSTITUTED PHENETHYLAMINE DERIVATIVES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2001-10-31 EP disclosed