SCHEMBL4010060

SCHEMBL4010060

CCc1nc(-c2ccc(C)cc2)nc(C(C)C)c1OC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 5/20 0.36
DPP9 Q86TI2 4/20 0.36
DPP8 Q6V1X1 3/20 0.36
ADORA3 P0DMS8 3/20 0.36
ADORA1 P30542 1/20 0.36
NPC1 O15118 1/20 0.36
XBP1 P17861 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAPT P10636 2/20 0.36
PRNP P04156 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GCGR P47871 1/20 0.35
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
LIPE Q05469 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4011472 0.89 MAPT (0.39) ADORA3NPC1RAB9AATMNPSR1
SCHEMBL4011273 0.89 ADORA3 (0.38) DPP4DPP9DPP8ADORA3ADORA1
SCHEMBL4011136 0.86 RAB9A (0.38) HTTRAB9ANPSR1MAPTPRNP
SCHEMBL4009025 0.82 ACP1 (0.38) ADORA3ADORA1NPC1MAPTTSHR
SCHEMBL4010057 0.81 DPP4 (0.48) DPP4DPP9DPP8ADORA3ADORA1
SCHEMBL4009391 0.80 ALDH1A1 (0.41) DPP4DPP9ADORA3ADORA1HTT
SCHEMBL4007725 0.78 ADORA3 (0.39) ADORA3NPC1HTTRAB9ANPSR1
SCHEMBL4005144 0.78 PPARA (0.39) ADORA3NPC1RAB9AMAPTGABRA2
SCHEMBL4010068 0.78 PPARG (0.40) ADORA3RAB9AATMNPSR1MAPT
SCHEMBL8038540 0.78 GCGR (0.45) DPP4DPP9DPP8ADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080248-A1 SUBSTITUTED 2-PHENYLPYRIMIDINE-5-CARBOXYLIC ACIDS AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed