SCHEMBL4012559

SCHEMBL4012559

CC(C)(O)c1ncnc2c1c(-c1cccc(Cl)c1Cl)cn2CC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 5/20 0.40
MCL1 Q07820 2/20 0.35
P2RX7 Q99572 4/20 0.32
FLT3 P36888 1/20 0.32
EIF2AK3 Q9NZJ5 1/20 0.32
KMO O15229 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
CFD P00746 1/20 0.31
PDGFRB P09619 1/20 0.31
FGFR1 P11362 1/20 0.31
SRC P12931 1/20 0.31
PDGFRA P16234 1/20 0.31
PDK1 Q15118 1/20 0.31
PDK2 Q15119 1/20 0.31
PDK3 Q15120 1/20 0.31
PDK4 Q16654 1/20 0.31
MAPK14 Q16539 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13769680 0.87 MAPK14 (0.40) CCR4P2RX7EIF2AK3MAPK14
SCHEMBL4008416 0.85 CCR4 (0.39) CCR4MCL1P2RX7EIF2AK3KMO
SCHEMBL4013000 0.83 CCR4 (0.39) CCR4MCL1P2RX7KMOPTGDR2
SCHEMBL4009501 0.76 SCN9A (0.36) CCR4P2RX7EIF2AK3SRC
SCHEMBL4007615 0.75 SRC (0.43) CCR4MCL1P2RX7SRC
SCHEMBL4007097 0.74 ALOX15 (0.36) CCR4MCL1PTGDR2SRC
SCHEMBL4014280 0.74 EGLN1 (0.34) CCR4MCL1P2RX7PTGDR2SRC
SCHEMBL13769710 0.74 KCNH2 (0.40)
SCHEMBL13769716 0.74 CALCRL (0.56)
SCHEMBL4008754 0.73 FLT4 (0.44) CCR4MCL1EIF2AK3SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed