SCHEMBL4022798

SCHEMBL4022798

CC1NC(=O)C(c2ccc(C#N)cc2)=C([C@H]2CC[C@@H](C(F)(F)F)CC2)N1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.37
KIF11 P52732 2/20 0.33
ACACB O00763 1/20 0.31
ACACA Q13085 1/20 0.31
PTPN5 P54829 1/20 0.31
KCNH2 Q12809 2/20 0.31
HRH3 Q9Y5N1 1/20 0.31
DRD2 P14416 2/20 0.30
DRD4 P21917 2/20 0.30
DRD3 P35462 2/20 0.30
ELANE P08246 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4756695 0.68 HSD11B1 (0.39) HSD11B1
SCHEMBL13746898 0.68 HSD11B1 (0.39) HSD11B1
SCHEMBL4755201 0.65 HSD11B1 (0.38) HSD11B1
SCHEMBL4755140 0.63 HSD11B1 (0.38) HSD11B1
SCHEMBL30429836 0.59 PDK1 (0.59) HSD11B1KCNH2CYP2C9
SCHEMBL16441196 0.58 KIF11 (0.62) KIF11PTPN5KCNH2
SCHEMBL1087536 0.58 NOTUM (0.42) KIF11
SCHEMBL14649680 0.58 HRH3 (0.54) HSD11B1KIF11KCNH2HRH3
SCHEMBL11524401 0.58 HRH3 (0.54) HSD11B1KIF11KCNH2HRH3
SCHEMBL11524397 0.58 HRH3 (0.54) HSD11B1KIF11KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed