SCHEMBL4029596

SCHEMBL4029596

CN(Cc1cc(Br)c(S(=O)(=O)c2cccc(F)c2)s1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 10/20 0.37
ABCC9 O60706 1/20 0.35
ABCC8 Q09428 1/20 0.35
KCNJ11 Q14654 1/20 0.35
KCNJ8 Q15842 1/20 0.35
CLK1 P49759 1/20 0.35
CLK2 P49760 1/20 0.35
DYRK1A Q13627 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
RIPK1 Q13546 1/20 0.34
GLS O94925 1/20 0.34
IDH1 O75874 1/20 0.34
KMT2A Q03164 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654644 0.89 HTR2C (0.38) GLSKMT2AHTR2CSLC6A4
SCHEMBL3651795 0.87 MEP1B (0.38) ABCC9ABCC8KCNJ11KCNJ8CLK1
Carbamic Acid SCHEMBL3651234 0.86 HTR2C (0.37) GLSKMT2AHTR2CSLC6A4
SCHEMBL4129164 0.86 HTR6 (0.38) HTR6KMT2A
SCHEMBL3652101 0.82 KAT6A (0.36) ABCC9ABCC8KCNJ11KCNJ8CLK1
SCHEMBL4029601 0.79 ABCC9 (0.36) HTR6ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL3654959 0.77 AR (0.36) CLK1CLK2DYRK1ACLK4DYRK1B
Hydrochloric Acid SCHEMBL3654116 0.76 HTR6 (0.35) HTR6GLSHTR2AHTR2C
SCHEMBL22013593 0.75 CACNA1G (0.36) RIPK1GLSHTR2AHTR2CSLC6A4
SCHEMBL3647494 0.75 GLS (0.35) GLSHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed