SCHEMBL4037774

SCHEMBL4037774

CCc1noc(-c2ccc(CCl)cc2)c1N(C(=O)O)C(c1ccccc1)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 1/20 0.33
S1PR1 P21453 5/20 0.32
HDAC4 P56524 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC7 Q8WUI4 2/20 0.32
HDAC5 Q9UQL6 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC2 Q92769 1/20 0.32
S1PR3 Q99500 3/20 0.31
HDAC9 Q9UKV0 1/20 0.31
TRPV1 Q8NER1 2/20 0.31
MLYCD O95822 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PTPN1 P18031 1/20 0.31
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030341 0.88 LPAR1 (0.39) LPAR1S1PR1HDAC4HDAC6HDAC1
SCHEMBL4034923 0.80 MEN1 (0.34) LPAR1S1PR1S1PR3L3MBTL1PPARG
SCHEMBL4029487 0.73 LPAR1 (0.48) LPAR1S1PR1TRPV1MLYCDL3MBTL1
SCHEMBL4031683 0.73 TRPA1 (0.43) LPAR1S1PR3MLYCD
SCHEMBL4034622 0.69 LPAR1 (0.38) LPAR1PTPN1PPARGPPARALMNA
SCHEMBL16060790 0.69 POLB (0.38) LPAR1S1PR1HDAC6HDAC1HDAC3
SCHEMBL4035140 0.69 KMT2A (0.44) MAPTNPSR1NPC1
SCHEMBL4033264 0.68 LPAR1 (0.40) LPAR1S1PR1HDAC6HDAC1HDAC3
SCHEMBL4033611 0.68 LPAR1 (0.40) LPAR1MAPTNPC1RAB9A
SCHEMBL4034499 0.67 LPAR1 (0.48) LPAR1S1PR1HDAC6HDAC1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed