SCHEMBL4035480

SCHEMBL4035480

O=Cc1ccc(-c2ccccc2)c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
CSNK2A1 P68400 2/20 0.49
CYP2A6 P11509 2/20 0.48
ALDH1A3 P47895 3/20 0.47
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
VCAM1 P19320 1/20 0.41
ALDH3A1 P30838 2/20 0.40
DRD1 P21728 2/20 0.40
HSD17B10 Q99714 1/20 0.40
IP6K1 Q92551 1/20 0.40
CTRC Q99895 2/20 0.39
TRIM24 O15164 1/20 0.39
TRIM33 Q9UPN9 1/20 0.39
PTPN11 Q06124 1/20 0.37
ESR1 P03372 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30185446 1.00 ALDH1A1 (0.55) ALDH1A1CSNK2A1CYP2A6ALDH1A3KDM4E
SCHEMBL30185447 1.00 ALDH1A1 (0.55) ALDH1A1CSNK2A1CYP2A6ALDH1A3KDM4E
SCHEMBL13638172 0.87 ALDH1A1 (0.53) ALDH1A1ALDH1A3MEN1NPC1KMT2A
SCHEMBL8176964 0.85 ALDH1A1 (0.55) ALDH1A1CSNK2A1CYP2A6ALDH1A3KDM4E
SCHEMBL30679643 0.84 ALDH1A1 (0.50) ALDH1A1ALDH1A3MEN1NPC1KMT2A
SCHEMBL35967 0.82 ALDH1A1 (0.48) ALDH1A1CYP2A6KDM4EMEN1NPC1
SCHEMBL4887408 0.81 ALDH5A1 (0.52) ALDH1A1ALDH1A3KDM4EVCAM1HSD17B10
SCHEMBL25613984 0.81 ALDH1A1 (0.55) ALDH1A1ALDH1A3MEN1KMT2AVCAM1
SCHEMBL8759091 0.81 CSNK2A1 (0.49) ALDH1A1CSNK2A1CYP2A6NPC1HSD17B10
SCHEMBL5490742 0.78 ALDH1A1 (0.50) ALDH1A1CYP2A6KDM4EMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1075480-A4 PURIFICATION OF CARBOXALDEHYDE LILLY CO ELI (US) 2002-01-23 EP claimed
EP-1075480-A1 PURIFICATION OF CARBOXALDEHYDE ELI LILLY AND COMPANY (US) 2001-02-14 EP claimed
WO-1999057123-A1 PURIFICATION OF CARBOXALDEHYDE ELI LILLY AND COMPANY (US) 1999-11-11 WO claimed
US-20260070901-A1 NOVEL COMPOUNDS AS CK2 INHIBITORS CAMBRIDGE ENTPR LTD (GB) 2026-03-12 US disclosed
EP-4584267-A1 NOVEL COMPOUNDS AS CK2 INHIBITORS Cambridge Enterprise Limited (GB) 2025-07-16 EP disclosed
US-20240287060-A1 BENZO[C][2,6]NAPHTHYRIDINE DERIVATIVES, COMPOSITIONS AND THERAPEUTIC USES THEREOF CAMBRIDGE ENTERPRISE LIMITED (GB) 2024-08-29 US disclosed
WO-2024052692-A1 NOVEL COMPOUNDS AS CK2 INHIBITORS CAMBRIDGE ENTERPRISE LIMITED (GB) 2024-03-14 WO disclosed
EP-4301752-A1 BENZO[C][2,6]NAPHTHYRIDINE DERIVATIVES, COMPOSITIONS AND THERAPEUTIC USES THEREOF Cambridge Enterprise Limited (GB) 2024-01-10 EP disclosed
US-11866436-B2 Benzo[c][2,6]naphthyridine derivatives, compositions and therapeutic uses thereof CAMBRIDGE ENTERPRISE LIMITED (GB) 2024-01-09 US disclosed
CN-117295736-A Benzo [ C ] [2,6] naphthyridine derivatives, compositions thereof and therapeutic uses thereof 剑桥实业有限公司 2023-12-26 CN disclosed
US-20230250097-A1 BENZO[C][2,6]NAPHTHYRIDINE DERIVATIVES, COMPOSITIONS AND THERAPEUTIC USES THEREOF Apollo Therapeutics Limited (GB) 2023-08-10 US disclosed
EP-1501509-A4 ARYL-LINK-ARYL SUBSTITUTED THIAZOLIDINE-DIONE AND OXAZOLIDINE-DIONE AS SODIUM CHANNEL BLOCKERS MERCK & CO INC (US) 2009-07-15 EP disclosed
CN-1960969-A Histamine H3 receptor agents, methods of preparation and therapeutic uses thereof LILLY CO ELI (US) 2007-05-09 CN disclosed
EP-1501509-A2 ARYL-LINK-ARYL SUBSTITUTED THIAZOLIDINE-DIONE AND OXAZOLIDINE-DIONE AS SODIUM CHANNEL BLOCKERS Merck & Co., Inc. (US) 2005-02-02 EP disclosed
WO-2004024061-A2 ARYL-LINK-ARYL SUBSTITUTED THIAZOLIDINE-DIONE AND OXAZOLIDINE-DIONE AS SODIUM CHANNEL BLOCKERS MERCK & CO., INC. (US) 2004-03-25 WO disclosed
EP-1075480-A4 PURIFICATION OF CARBOXALDEHYDE LILLY CO ELI (US) 2002-01-23 EP disclosed
EP-1075480-A1 PURIFICATION OF CARBOXALDEHYDE ELI LILLY AND COMPANY (US) 2001-02-14 EP disclosed
WO-1999057123-A1 PURIFICATION OF CARBOXALDEHYDE ELI LILLY AND COMPANY (US) 1999-11-11 WO disclosed
US-3966801-A ANTIINFLAMMATORY AGENTS WILLIAM H. RORER, INC. (US) 1976-06-29 US disclosed
US-3950427-A ANTIINFLAMMATORY, ANTIPYRETIC BOEHRINGER INGELHEIM GMBH (DT) 1976-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230250097-A1 BENZO[C][2,6]NAPHTHYRIDINE DERIVATIVES, COMPOSITIONS AND THERAPEUTIC USES THEREOF CSNK1A1, CSNK1D, CSNK2A1 ALDH1A1 2913/4885CSNK2A1 3/4885CYP2A6 1259/4885
US-11866436-B2 Benzo[c][2,6]naphthyridine derivatives, compositions and therapeutic uses thereof ABCB11, CEL, NDC1 ALDH1A1 681/4885CSNK2A1 517/4885CYP2A6 113/4885
US-20240287060-A1 BENZO[C][2,6]NAPHTHYRIDINE DERIVATIVES, COMPOSITIONS AND THERAPEUTIC USES THEREOF CSNK1A1, CSNK1D, CSNK2A1 ALDH1A1 2913/4885CSNK2A1 3/4885CYP2A6 1259/4885
US-20260070901-A1 NOVEL COMPOUNDS AS CK2 INHIBITORS CSNK1A1, CSNK2A3, CSNK1G1 ALDH1A1 3874/4885CSNK2A1 5/4885CYP2A6 2977/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.