SCHEMBL4039235

SCHEMBL4039235

C[C@@](O)(Cc1c[nH]c2ccccc12)NC(=O)c1cccc(C#CCCCO)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.44
EPHX2 P34913 1/20 0.44
CDK4 P11802 3/20 0.41
CCND1 P24385 3/20 0.41
MEN1 O00255 6/20 0.40
KMT2A Q03164 6/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
ADRB3 P13945 1/20 0.37
GPR84 Q9NQS5 3/20 0.37
MAPT P10636 1/20 0.37
NMBR P28336 1/20 0.37
ANO1 Q5XXA6 1/20 0.37
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028879 0.91 ALOX5 (0.47) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL4034817 0.85 ALOX5 (0.46) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL4034576 0.80 ALOX5 (0.52) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL3941237 0.79 ALOX5 (0.47) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL4029965 0.79 CDK4 (0.47) CDK4CCND1MEN1KMT2ANPC1
SCHEMBL3944233 0.77 ALOX5 (0.46) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL4035462 0.76 KMT2A (0.41) MEN1KMT2AMAPTNMBRCYP2D6
SCHEMBL4632724 0.75 GPR84 (0.40) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL4039237 0.75 ALOX5 (0.44) ALOX5EPHX2CDK4CCND1MEN1
SCHEMBL4039229 0.75 ALOX5 (0.44) ALOX5EPHX2CDK4CCND1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed