SCHEMBL4034576

SCHEMBL4034576

CCC(C#Cc1cccc(C(=O)N[C@](C)(O)Cc2c[nH]c3ccccc23)c1)C(N)=O

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.52
EPHX2 P34913 3/20 0.52
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
CDK4 P11802 1/20 0.39
CCND1 P24385 1/20 0.39
HPGDS O60760 2/20 0.38
TACR1 P25103 4/20 0.38
NMBR P28336 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ERAP2 Q6P179 2/20 0.37
CYP2D6 P10635 1/20 0.37
IL1RN P18510 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
CTSL P07711 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4028879 0.83 ALOX5 (0.47) ALOX5EPHX2MEN1KMT2ACDK4
SCHEMBL4034817 0.81 ALOX5 (0.46) ALOX5EPHX2MEN1KMT2ACDK4
SCHEMBL4039235 0.80 ALOX5 (0.44) ALOX5EPHX2MEN1KMT2ACDK4
SCHEMBL4029965 0.77 CDK4 (0.47) MEN1KMT2ACDK4CCND1NMBR
SCHEMBL4632724 0.75 GPR84 (0.40) ALOX5EPHX2MEN1KMT2ACDK4
SCHEMBL4038448 0.68 KMT2A (0.42) MEN1KMT2ATACR1NMBRKDM4E
SCHEMBL11829083 0.67 MEN1 (0.55) MEN1KMT2ACDK4CCND1TACR1
SCHEMBL4035462 0.66 KMT2A (0.41) MEN1KMT2ATACR1NMBRKDM4E
SCHEMBL5149351 0.66 ANO1 (0.41) MEN1KMT2ATACR1KDM4ECYP2D6
SCHEMBL4737661 0.65 ERAP2 (0.52) ALOX5EPHX2MEN1KMT2ACDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed