SCHEMBL4042300

SCHEMBL4042300

COc1ccc2oc(OC(=O)NC(CC(C)C)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)c3cccc[n+]3[O-])cc2c1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.37
TAS1R3 Q7RTX0 4/20 0.36
TAS1R1 Q7RTX1 4/20 0.36
CTSL P07711 9/20 0.33
CTSS P25774 6/20 0.33
CTSB P07858 5/20 0.33
CTSV O60911 2/20 0.33
HDAC8 Q9BY41 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045162 0.93 TAS1R3 (0.34) CTSKTAS1R3TAS1R1
SCHEMBL4043929 0.93 CTSV (0.32) CTSKTAS1R3TAS1R1CTSLCTSS
SCHEMBL4041781 0.92 CTSK (0.39) CTSKTAS1R3TAS1R1CTSLCTSS
SCHEMBL4043593 0.90 USP2 (0.33) CTSKTAS1R3TAS1R1
SCHEMBL4042354 0.90 TAS1R3 (0.37) CTSKTAS1R3TAS1R1CTSLCTSS
SCHEMBL4046540 0.88 CTSK (0.37) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4041991 0.86 CTSK (0.46) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4047816 0.85 CTSK (0.33) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4047148 0.84 CHRNB2 (0.39) CTSKTAS1R3TAS1R1CTSLCTSS
SCHEMBL4044439 0.84 CTSK (0.41) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed