SCHEMBL4043393

SCHEMBL4043393

CCCC(NC(=O)Oc1ccc(-c2ccccc2)s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
SMYD3 Q9H7B4 2/20 0.33
CTSK P43235 3/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
MMP13 P45452 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043813 0.93 CHRNB2 (0.36) FKBP1ACHRNB2CHRNA7CHRNA4SMYD3
SCHEMBL4044003 0.93 CTSK (0.40) FKBP1ACHRNB2CHRNA7CHRNA4CTSK
SCHEMBL4039018 0.90 HSD17B10 (0.36) CHRNB2CHRNA7CHRNA4CTSKCTSS
SCHEMBL4043998 0.89 FKBP1A (0.37) FKBP1ACHRNA7SMYD3CTSKCTSB
SCHEMBL4040719 0.88 SMYD3 (0.35) FKBP1ASMYD3CTSKCTSBCTSS
SCHEMBL4044808 0.88 CTSK (0.36) CHRNB2CHRNA7CHRNA4CTSKCTSS
SCHEMBL4044090 0.88 CTSK (0.34) CTSKMMP13
SCHEMBL4050153 0.88 SMYD3 (0.35) FKBP1ASMYD3
SCHEMBL4044586 0.87 CTSK (0.37) CHRNB2CHRNA7CHRNA4CTSKCTSS
SCHEMBL4042582 0.87 CTSK (0.44) FKBP1ACTSKCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed