SCHEMBL4043722

SCHEMBL4043722

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1ccccn1)Oc1cccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.40
CTSL P07711 4/20 0.36
CTSS P25774 4/20 0.36
MC4R P32245 1/20 0.36
MC3R P41968 1/20 0.36
MC1R Q01726 1/20 0.36
CTSB P07858 1/20 0.35
FNTA P49354 1/20 0.35
FNTB P49356 1/20 0.35
GRIA1 P42261 1/20 0.34
ACE2 Q9BYF1 1/20 0.34
TGM2 P21980 2/20 0.33
F12 P00748 1/20 0.33
ACE P12821 1/20 0.33
PTGS2 P35354 1/20 0.32
CASP1 P29466 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PSMB5 P28074 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049994 0.93 CTSK (0.40) CTSKCTSLCTSSMC4RMC3R
SCHEMBL6210598 0.89 CTSL (0.45) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4044603 0.88 MC4R (0.37) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4043883 0.87 CTSK (0.42) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4044768 0.86 CTSL (0.44) CTSKCTSLCTSSCTSB
SCHEMBL4045047 0.84 CTSL (0.37) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4046533 0.84 MAPK1 (0.36) CTSKCTSSMC4RMC3RMC1R
SCHEMBL4052754 0.82 CTSK (0.42) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4040381 0.82 MC4R (0.36) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4045030 0.81 CTSK (0.41) CTSKCTSLCTSSMC4RMC3R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed