SCHEMBL4043883

SCHEMBL4043883

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1ccccn1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.42
CTSL P07711 2/20 0.37
CTSS P25774 2/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
ACE2 Q9BYF1 1/20 0.36
ACE P12821 2/20 0.35
GRIA1 P42261 1/20 0.35
PRCP P42785 1/20 0.34
TGM2 P21980 1/20 0.34
MC4R P32245 1/20 0.34
MC3R P41968 1/20 0.34
MC1R Q01726 1/20 0.34
PSMB5 P28074 1/20 0.34
GLP1R P43220 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA4 P13612 1/20 0.33
ITGB7 P26010 1/20 0.33
OPRD1 P41143 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041556 0.93 CTSK (0.43) CTSKCTSLCTSSPRCPITGB1
SCHEMBL4052754 0.93 CTSK (0.42) CTSKCTSLCTSSPRCPMC4R
SCHEMBL4045030 0.92 CTSK (0.41) CTSKCTSLCTSSFNTAFNTB
SCHEMBL4044814 0.88 FNTA (0.35) CTSKFNTAFNTBACE2GRIA1
SCHEMBL4045333 0.88 CTSK (0.53) CTSKCTSLCTSS
SCHEMBL4045843 0.87 CTSK (0.43) CTSKCTSLCTSSTGM2
SCHEMBL4043722 0.87 CTSK (0.40) CTSKCTSLCTSSFNTAFNTB
SCHEMBL4049994 0.86 CTSK (0.40) CTSKCTSLCTSSFNTAFNTB
SCHEMBL4041003 0.85 CTSL (0.39) CTSKCTSLCTSS
SCHEMBL4044539 0.84 ITGA4 (0.36) CTSKCTSLCTSSFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed