SCHEMBL4045030

SCHEMBL4045030

O=C(NC(Cc1cccc(O)c1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1ccccn1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 4/20 0.41
CTSL P07711 2/20 0.37
CTSS P25774 2/20 0.37
TGM2 P21980 1/20 0.34
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
HPGDS O60760 1/20 0.33
MC4R P32245 1/20 0.33
MC3R P41968 1/20 0.33
MC1R Q01726 1/20 0.33
HTRA1 Q92743 3/20 0.33
PSMB5 P28074 1/20 0.33
GPR132 Q9UNW8 1/20 0.33
ITGB3 P05106 1/20 0.32
ITGAV P06756 1/20 0.32
KLKB1 P03952 1/20 0.32
MGLL Q99685 1/20 0.32
ACE P12821 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043883 0.92 CTSK (0.42) CTSKCTSLCTSSTGM2FNTA
SCHEMBL4041556 0.89 CTSK (0.43) CTSKCTSLCTSSHTRA1ITGB3
SCHEMBL4052754 0.89 CTSK (0.42) CTSKCTSLCTSSMC4RMC3R
SCHEMBL4043350 0.89 HTRA1 (0.35) CTSKCTSLCTSSFNTAFNTB
SCHEMBL4051296 0.86 CTSL (0.39) CTSKCTSLCTSS
SCHEMBL4045333 0.86 CTSK (0.53) CTSKCTSLCTSSMEN1KMT2A
SCHEMBL4045843 0.85 CTSK (0.43) CTSKCTSLCTSSTGM2MEN1
SCHEMBL4042165 0.85 EPHX1 (0.37) CTSKCTSLCTSSGPR132ACE
SCHEMBL4046932 0.84 GPR132 (0.35) CTSKCTSLCTSSFNTAFNTB
SCHEMBL4045091 0.82 CTSK (0.61) CTSKCTSLCTSSHPGDSMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed