SCHEMBL4043944

SCHEMBL4043944

O=C(NC(Cc1cccs1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)Oc1cc2sccc2s1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.33
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
PAX8 Q06710 1/20 0.31
ACE P12821 2/20 0.31
CHRNA7 P36544 1/20 0.31
CYP51A1 Q16850 1/20 0.30
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051435 0.90 HTRA1 (0.33) CTSKCTSSPAX8
SCHEMBL4042884 0.90 CTSK (0.41) CTSKCTSBCTSSPAX8ALDH1A1
SCHEMBL4038641 0.90 CTSK (0.33) CTSKPAX8ALDH1A1L3MBTL1
SCHEMBL4045954 0.88 SMYD3 (0.33) CTSKCTSBCTSSACECHRNA7
SCHEMBL4039560 0.86 HCRTR2 (0.33) CTSKCTSBCTSS
SCHEMBL4052028 0.84 CTSK (0.32) CTSKALDH1A1
SCHEMBL4040702 0.83 CTSK (0.38) CTSKCTSBCTSS
SCHEMBL4044961 0.82 CHRNB2 (0.35) CTSKCTSBCTSSPAX8ACE
SCHEMBL4044847 0.82 CHRNB2 (0.39) CTSKCTSBCTSSCHRNA7ALDH1A1
SCHEMBL4038998 0.81 CTSK (0.44) CTSKCTSBCTSSPAX8CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed