SCHEMBL404482

SCHEMBL404482

N#Cc1ccc(F)cc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TRPV4 Q9HBA0 1/20 0.42
KDM4E B2RXH2 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
CYP11B2 P19099 4/20 0.40
CYP11B1 P15538 3/20 0.40
USP2 O75604 1/20 0.38
AR P10275 1/20 0.38
KHK P50053 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CSNK2A1 P68400 1/20 0.36
KEAP1 Q14145 1/20 0.36
CUL4A Q13619 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
MPO P05164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12733363 0.84 CYP11B2 (0.54) ALDH1A1KDM4EMEN1KMT2AMAOA
SCHEMBL168901 0.82 ALDH1A1 (0.50) ALDH1A1TRPV4KDM4EMEN1KMT2A
SCHEMBL30262619 0.82 ALDH1A1 (0.50) ALDH1A1TRPV4KDM4EMEN1KMT2A
SCHEMBL573864 0.78 MAOB (0.53) ALDH1A1TRPV4KDM4EMAOAMAOB
SCHEMBL29137845 0.77 ALDH1A1 (0.44) ALDH1A1KEAP1GAAHTT
SCHEMBL9327450 0.77 ALDH1A1 (0.44) ALDH1A1KEAP1GAAHTT
SCHEMBL5070146 0.76 MEN1 (0.48) ALDH1A1TRPV4KDM4EMEN1KMT2A
SCHEMBL21131569 0.76 TRPV4 (0.45) ALDH1A1TRPV4KDM4EMEN1KMT2A
SCHEMBL2028221 0.76 KDM4E (0.55) ALDH1A1TRPV4KDM4EMEN1KMT2A
SCHEMBL57346 0.76 TRPV4 (0.61) ALDH1A1TRPV4MAOAMAOBCYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 253 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332789-A Preparation method of 4-amino-2-fluorobenzamide 上海康鹏科技股份有限公司 2023-06-27 CN claimed
CN-106946800-A A kind of synthetic method of (1H, the 3H) diketone of quinazoline 2,4 and its derivative 华东师范大学 2017-07-14 CN claimed
US-12528816-B2 Substituted imidazo [1,2-b] pyridazines and [1, 2, 4] triazolo [ 4,3-b] pyridazines as camkii inhibitors CARDURION PHARMACEUTICALS, INC. (US) 2026-01-20 US disclosed
EP-4660186-A1 ACID ADDITION SALT OF 4-AMINO-2-HALOBENZONITRILE COMPOUND AND METHOD FOR PRODUCING SAME SUGAI CHEMICAL INDUSTRY CO., LTD. (JP) 2025-12-10 EP disclosed
EP-4635568-A2 COMPOUNDS, SALTS THEREOF AND METHODS FOR TREATMENT OF DISEASES ACADIA Pharmaceuticals Inc. (US) 2025-10-22 EP disclosed
EP-3672954-B1 COMPOUNDS, SALTS THEREOF AND THEIR USE FOR THE TREATMENT OF DISEASES ACADIA PHARM INC (US) 2025-08-13 EP disclosed
US-20250197385-A1 COMPOUNDS, SALTS THEREOF AND METHODS FOR TREATMENT OF DISEASES ACADIA PHARM INC (US) 2025-06-19 US disclosed
US-20250179072-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2025-06-05 US disclosed
CN-119768407-A Protein phosphatase agonist and application thereof 南京中瑞药业有限公司 2025-04-04 CN disclosed
CN-116102495-B 1,2,3, 4-Tetrahydro-9-aminoacridine compound and application thereof 浙江工业大学 2025-03-21 CN disclosed
CN-119331429-A Azo red dye compound and preparation method and application thereof 南京晓庄学院 2025-01-21 CN disclosed
US-5206387-A Chemical intermediates for memory enhancing drugs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-04-27 US disclosed
US-5189054-A 3-amidoindolyl derivatives and pharmaceutical compositions thereof MERRELL DOW PHARMACEUTICALS INC. (US) 1993-02-23 US disclosed
US-5112830-A Cognition Activators HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1992-05-12 US disclosed
EP-0483881-A1 3-Amidoindolyl derivatives MERRELL PHARMACEUTICALS INC. (US) 1992-05-06 EP disclosed
US-5002955-A Pyrroloquinolines for enhancement of memory HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-03-26 US disclosed
EP-0371388-A2 Acridine derivatives FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-06-06 EP disclosed
US-4843079-A ALZHEIMER*S DISEASE HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-27 US disclosed
EP-0287977-A2 Fused heteroalkylene quinolinamines, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1988-10-26 EP disclosed
EP-0268871-A1 Quinoline derivatives SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1988-06-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12528816-B2 Substituted imidazo [1,2-b] pyridazines and [1, 2, 4] triazolo [ 4,3-b] pyridazines as camkii inhibitors RYR2, CACNA1C, CAMK4 ALDH1A1 1793/4885TRPV4 788/4885KDM4E 4364/4885
US-20250179072-A1 TRICYCLIC AKR1C3 DEPENDENT KARS INHIBITORS AKR1C2, AKR1B1, AKR1C1 ALDH1A1 234/4885TRPV4 3597/4885KDM4E 1460/4885
US-20250197385-A1 COMPOUNDS, SALTS THEREOF AND METHODS FOR TREATMENT OF DISEASES SLC10A1, CYP27A1, CYP11B2 ALDH1A1 240/4885TRPV4 3467/4885KDM4E 4595/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.