SCHEMBL4046652

SCHEMBL4046652

CCCC(NC(=O)Oc1ccc2ccccc2n1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.35
CHRNA7 P36544 2/20 0.35
CHRNA4 P43681 2/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
FKBP1A P62942 1/20 0.34
PREP P48147 1/20 0.34
FAP Q12884 1/20 0.34
SMYD3 Q9H7B4 2/20 0.33
CTSB P07858 2/20 0.33
CTSS P25774 2/20 0.33
CTSK P43235 2/20 0.33
CTSL P07711 1/20 0.33
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
TSHR P16473 1/20 0.32
MC4R P32245 1/20 0.32
MC3R P41968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051166 0.93 CTSK (0.39) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3
SCHEMBL4045110 0.92 PREP (0.35) FKBP1APREPFAPSMYD3CTSB
SCHEMBL4048207 0.90 HSD17B10 (0.36) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3
SCHEMBL4047844 0.89 SMYD3 (0.35) FKBP1ASMYD3CTSKMC4RMC3R
SCHEMBL6211183 0.89 CTSK (0.42) CHRNB2CHRNA7CHRNA4PREPFAP
SCHEMBL4045687 0.88 MC4R (0.34) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3
SCHEMBL4044622 0.88 CTSK (0.38) PREPFAPCTSBCTSSCTSK
SCHEMBL4041238 0.87 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4CHRNB4CHRNA3
SCHEMBL4040719 0.87 SMYD3 (0.35) FKBP1APREPFAPSMYD3CTSB
SCHEMBL4043998 0.86 FKBP1A (0.37) CHRNA7FKBP1ASMYD3CTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed