SCHEMBL4045110

SCHEMBL4045110

CCCC(NC(=O)Oc1cnc2ccccc2n1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
SMYD3 Q9H7B4 2/20 0.35
FKBP1A P62942 1/20 0.34
POLB P06746 1/20 0.33
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
TSHR P16473 1/20 0.32
CTSK P43235 2/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046952 0.93 CTSK (0.39) SMYD3FKBP1ACTSKCTSBCTSS
SCHEMBL4046652 0.92 CHRNB2 (0.35) PREPFAPSMYD3FKBP1ACYP2C9
SCHEMBL4046666 0.90 HSD17B10 (0.36) PREPFAPSMYD3ALDH1A1TSHR
SCHEMBL4042075 0.89 PREP (0.36) PREPFAPCTSKCTSBCTSS
SCHEMBL4050283 0.88 PREP (0.35) PREPFAPCTSKCTSS
SCHEMBL4045929 0.87 PREP (0.36) PREPFAPPOLBCTSK
SCHEMBL4047844 0.87 SMYD3 (0.35) SMYD3FKBP1ACTSK
SCHEMBL4043998 0.86 FKBP1A (0.37) SMYD3FKBP1ACTSKCTSBCTSS
SCHEMBL4045549 0.86 CTSL (0.39) PREPFAPCTSKCTSBCTSS
SCHEMBL4047431 0.86 ALDH1A1 (0.37) PREPFAPSMYD3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed