SCHEMBL4047338

SCHEMBL4047338

COc1ccc2oc(OC(=O)NC3(C(=O)N4CCC5C4C(=O)CN5S(=O)(=O)c4cccc[n+]4[O-])CCCCC3)cc2c1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 1/20 0.33
FAAH O00519 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
RECQL P46063 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALDH1A1 P00352 2/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP3 P08254 1/20 0.30
MMP7 P09237 1/20 0.30
MMP9 P14780 1/20 0.30
MMP8 P22894 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044715 0.90 MMP1 (0.34) TACR2FAAHTRPV1KDM4EMEN1
SCHEMBL4050955 0.86 CTSK (0.37) FAAHTRPV1
SCHEMBL4045182 0.84 KCNQ1 (0.37) KDM4EMEN1CYP1A2RECQLKMT2A
SCHEMBL4050428 0.83 HPGD (0.33) TACR2FAAHTRPV1KDM4EMEN1
SCHEMBL4040665 0.83 HPGD (0.38) TACR2FAAHTRPV1KDM4EMEN1
SCHEMBL4042300 0.82 CTSK (0.37)
SCHEMBL4043929 0.82 CTSV (0.32)
SCHEMBL4045162 0.82 TAS1R3 (0.34)
SCHEMBL4046100 0.81 KLK7 (0.35) TACR2FAAHTRPV1KDM4EMEN1
SCHEMBL4042598 0.81 CTSK (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1662876-A4 NOVEL CRYSTALLINE FORMS OF A PHOSPHORIC ACID SALT OF A DIPEPTIDYL PEPTIDASE-IV INHIBITOR MERCK & CO INC (US) 2009-01-14 EP claimed
JP-2007504230-A 2007-03-01 JP claimed
EP-1662876-A2 NOVEL CRYSTALLINE FORMS OF A PHOSPHORIC ACID SALT OF A DIPEPTIDYL PEPTIDASE-IV INHIBITOR Merck & Co., Inc. (US) 2006-06-07 EP claimed
WO-2005020920-A2 NOVEL CRYSTALLINE FORMS OF A PHOSPHORIC ACID SALT OF A DIPEPTIDYL PEPTIDASE-IV INHIBITOR MERCK & CO., INC. (US) 2005-03-10 WO claimed