SCHEMBL4050428

SCHEMBL4050428

COc1ccc2oc(OC(=O)NC3(C(=O)N4CCC5C4C(=O)CN5S(=O)(=O)C(=O)c4ccccn4)CCCCC3)cc2c1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.33
ALDH1A1 P00352 6/20 0.32
KDM4E B2RXH2 4/20 0.32
HSD17B10 Q99714 3/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
FAAH O00519 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
CYP1A2 P05177 1/20 0.32
RECQL P46063 1/20 0.32
TACR2 P21452 1/20 0.31
LMNA P02545 1/20 0.31
ADRB2 P07550 1/20 0.30
RAB9A P51151 1/20 0.30
GLA P06280 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050955 0.91 CTSK (0.37) HPGDFAAHTRPV1
SCHEMBL4047235 0.89 CTSL (0.36) HPGDALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL4046100 0.88 KLK7 (0.35) HPGDALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL4040665 0.88 HPGD (0.38) HPGDALDH1A1KDM4EHSD17B10FAAH
SCHEMBL4045182 0.85 KCNQ1 (0.37) HPGDALDH1A1KDM4EHSD17B10SMN1; SMN2
SCHEMBL4047338 0.83 TACR2 (0.33) ALDH1A1KDM4EHSD17B10FAAHTRPV1
SCHEMBL4044715 0.83 MMP1 (0.34) ALDH1A1KDM4EHSD17B10FAAHTRPV1
SCHEMBL4043466 0.83 CHRNB2 (0.40) HPGDALDH1A1KDM4EKMT2ATACR2
SCHEMBL4046667 0.83 CTSK (0.37) HPGD
SCHEMBL4050896 0.82 HPGD (0.34) HPGDALDH1A1KDM4EHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed