SCHEMBL4049366

SCHEMBL4049366

COc1ccc2oc(OC(=O)NC(CC(C)C)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)C(=O)c3cccnc3)cc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
TAS1R3 Q7RTX0 4/20 0.35
TAS1R1 Q7RTX1 4/20 0.35
ALDH1A1 P00352 3/20 0.35
HPGD P15428 1/20 0.35
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
BLM P54132 1/20 0.34
KMT2A Q03164 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
KLK7 P49862 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
NAMPT P43490 1/20 0.33
CTSL P07711 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043842 0.93 CHRNB2 (0.36) CTSKCHRNB2CHRNA7CHRNA4ALDH1A1
SCHEMBL4047814 0.93 CHRNB2 (0.36) CTSKCHRNB2CHRNA7CHRNA4TAS1R3
SCHEMBL4045633 0.92 CTSK (0.41) CTSKALDH1A1MAPTMMP1MMP3
SCHEMBL4047148 0.91 CHRNB2 (0.39) CTSKCHRNB2CHRNA7CHRNA4TAS1R3
SCHEMBL4045350 0.91 CHRNB2 (0.34) CTSKCHRNB2CHRNA7CHRNA4ALDH1A1
SCHEMBL4046703 0.89 CHRNB2 (0.42) CTSKCHRNB2CHRNA7CHRNA4TAS1R3
SCHEMBL4046667 0.88 CTSK (0.37) CTSKTAS1R3TAS1R1HPGDCTSL
SCHEMBL4043435 0.88 CTSK (0.38) CTSKCHRNB2CHRNA7CHRNA4ALDH1A1
SCHEMBL4043183 0.87 CTSK (0.43) CTSKALDH1A1MAPTMMP1MMP3
SCHEMBL4041991 0.85 CTSK (0.46) CTSKCTSLCTSSCTSVCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed