SCHEMBL4045350

SCHEMBL4045350

COc1ccc2oc(OC(=O)NC(Cc3cccs3)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)C(=O)c3cccnc3)cc2c1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
ALDH1A1 P00352 4/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
BLM P54132 1/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HPGD P15428 1/20 0.33
TRPM8 Q7Z2W7 2/20 0.32
F12 P00748 1/20 0.32
AVPR1B P47901 1/20 0.31
USP30 Q70CQ3 1/20 0.31
KLK7 P49862 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
NAMPT P43490 1/20 0.31
CTSK P43235 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043432 0.91 KCNQ1 (0.38) CHRNB2CHRNA7CHRNA4ALDH1A1MEN1
SCHEMBL4049366 0.91 CTSK (0.38) CHRNB2CHRNA7CHRNA4ALDH1A1MAPT
SCHEMBL4043842 0.90 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4ALDH1A1MAPT
SCHEMBL4047814 0.90 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4ALDH1A1MAPT
SCHEMBL4046322 0.90 CHRNB2 (0.38) CHRNB2CHRNA7CHRNA4ALDH1A1KMT2A
SCHEMBL4038978 0.89 USP30 (0.34) HPGDTRPM8USP30CTSK
SCHEMBL4049501 0.86 CTSK (0.40) HPGDTRPM8CTSK
SCHEMBL4044847 0.86 CHRNB2 (0.39) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4051635 0.85 HPGD (0.37) ALDH1A1L3MBTL1HPGDTRPM8USP30
SCHEMBL4044402 0.84 GAA (0.36) ALDH1A1TRPM8USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed